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Phieng Siliphaivanh

Discovery of a Novel ERK Inhibitor with Activity in Models of Acquired Resistance to BRAF and MEK Inhibitors
2013 · Erick J. Morris, Sharda Jha, et al. · Cancer Discovery · 664
Total Synthesis of Gypsetin, Deoxybrevianamide E, Brevianamide E, and Tryprostatin B: Novel Constructions of 2,3-Disubstituted Indoles
1999 · Jeffrey M. Schkeryantz, Jonathan C. G. Woo, et al. · Journal of the American Chemical Society · 182
Enantioselective Total Synthesis of (+)-Leucascandrolide A Macrolactone
2003 · Michael T. Crimmins, Phieng Siliphaivanh · Organic Letters · 69
Identification of Potent Reverse Indazole Inhibitors for HPK1
2021 · Elsie C. Yu, Joey L. Methot, et al. · ACS Medicinal Chemistry Letters · 47
Allosteric Modulation of Protein Arginine Methyltransferase 5 (PRMT5)
2020 · Rachel L. Palte, Sebastian E. Schneider, et al. · ACS Medicinal Chemistry Letters · 45
Design of novel histone deacetylase inhibitors
2007 · Phieng Siliphaivanh, Paul Harrington, et al. · Bioorganic & Medicinal Chemistry Letters · 42
The Discovery of Two Novel Classes of 5,5-Bicyclic Nucleoside-Derived PRMT5 Inhibitors for the Treatment of Cancer
2021 · Ryan V. Quiroz, Michael H. Reutershan, et al. · Journal of Medicinal Chemistry · 40
Discovery of 1-(1H-Pyrazolo[4,3-c]pyridin-6-yl)urea Inhibitors of Extracellular Signal-Regulated Kinase (ERK) for the Treatment of Cancers
2016 · Jongwon Lim, Elizabeth H. Kelley, et al. · Journal of Medicinal Chemistry · 40
Purine derivatives as potent γ-secretase modulators
2010 · Alexey Rivkin, Sean P. Ahearn, et al. · Bioorganic & Medicinal Chemistry Letters · 35
Delayed and Prolonged Histone Hyperacetylation with a Selective HDAC1/HDAC2 Inhibitor
2014 · Joey L. Methot, Dawn Mampreian Hoffman, et al. · ACS Medicinal Chemistry Letters · 34
Structure-Based Discovery of Proline-Derived Arginase Inhibitors with Improved Oral Bioavailability for Immuno-Oncology
2021 · Min Lu, Hongjun Zhang, et al. · ACS Medicinal Chemistry Letters · 32
Structural insights on ligand recognition at the human leukotriene B4 receptor 1
2021 · Nairie Michaelian, Anastasiia Sadybekov, et al. · Nature Communications · 23
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Phenylglycine and phenylalanine derivatives as potent and selective HDAC1 inhibitors (SHI-1)
2008 · Kevin J. Wilson, David J. Witter, et al. · Bioorganic & Medicinal Chemistry Letters · 23
Anti-inflammatory actions of Chemoattractant Receptor-homologous molecule expressed on Th2 by the antagonist MK-7246 in a novel rat model of Alternaria alternata elicited pulmonary inflammation
2014 · Malgorzata A. Gil, Michael Caniga, et al. · European Journal of Pharmacology · 11
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Discovery of MK-8318, a Potent and Selective CRTh2 Receptor Antagonist for the Treatment of Asthma
2018 · Xianhai Huang, Jason Brubaker, et al. · ACS Medicinal Chemistry Letters · 10
Label-Free, LC-MS-Based Assays to Quantitate Small-Molecule Antagonist Binding to the Mammalian BLT1 Receptor
2017 · Xun Chen, Steven Stout, et al. · SLAS DISCOVERY · 7
Quality by design (QbD) of amide isosteres: 5,5-Disubstituted isoxazolines as potent CRTh2 antagonists with favorable pharmacokinetic and drug-like properties
2014 · Dong Xiao, Xiaohong Zhu, et al. · Bioorganic & Medicinal Chemistry Letters · 7
The Discovery of Bridged Benzoazepine Amides as Selective Allosteric Modulators of RIPK1
2025 · Joanna L. Chen, Joey L. Methot, et al. · ACS Medicinal Chemistry Letters · 5
Supplementary Figure Legends from Discovery of a Novel ERK Inhibitor with Activity in Models of Acquired Resistance to BRAF and MEK Inhibitors
2023 · Erick J. Morris, Sharda Jha, et al.
Supplementary Figures from Discovery of a Novel ERK Inhibitor with Activity in Models of Acquired Resistance to BRAF and MEK Inhibitors
2023 · Erick J. Morris, Sharda Jha, et al.
Data from Discovery of a Novel ERK Inhibitor with Activity in Models of Acquired Resistance to BRAF and MEK Inhibitors
2023 · Erick J. Morris, Sharda Jha, et al.
Enantioselective Total Synthesis of (+)‐Leucascandrolide: A Macrolactone.
2004 · Michael T. Crimmins, Phieng Siliphaivanh · ChemInform
ChemInform Abstract: Total Synthesis of Gypsetin, Deoxybrevianamide E, Brevianamide E, and Tryprostatin B: Novel Constructions of 2,3‐Disubstituted Indoles.
2000 · Jeffrey M. Schkeryantz, Jonathan C.G. Woo, et al. · ChemInform
Works count: 24
Citation count: 1,316
H-index: 13
I10-index: 15
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