Author

Timothy M. Chapman

Institution: LifeArc

Observed institutions: LifeArc, University of Toronto, University of Oxford, Drexel University, Medical Research Council

ORCID: 0000-0002-7396-0569

Observed ORCID: 0000-0002-7396-0569

OpenAlex ID: A5034830599

Rhodium-Catalyzed Asymmetric Allylic Substitution with Boronic Acid Nucleophiles

2006 · Frederic Menard, Timothy M. Chapman, et al. · Organic Letters · 93

Glyco- and Peptidomimetics from Three-Component Joullié−Ugi Coupling Show Selective Antiviral Activity

2004 · Timothy M. Chapman, Ieuan G. Davies, et al. · Journal of the American Chemical Society · 86

Highly Diastereoselective Additions to Polyhydroxylated Pyrrolidine Cyclic Imines: Ready Elaboration of Aza‐Sugar Scaffolds To Create Diverse Carbohydrate‐Processing Enzyme Probes

2003 · Timothy M. Chapman, Steve Courtney, et al. · Chemistry - A European Journal · 86

Novel Cyclic Sugar Imines: Carbohydrate Mimics and Easily Elaborated Scaffolds for Aza-Sugars

2001 · Benjamin G. Davis, Michael A. T. Maughan, et al. · Organic Letters · 71

Recent advances in the design and development of formyl peptide receptor 2 (FPR2/ALX) agonists as pro-resolving agents with diverse therapeutic potential

2021 · Monika Maciuszek, Antonino Cacace, et al. · European Journal of Medicinal Chemistry · 63

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Substituted aminopyrimidine protein kinase B (PknB) inhibitors show activity against Mycobacterium tuberculosis

2012 · Timothy M. Chapman, Nathalie Bouloc, et al. · Bioorganic & Medicinal Chemistry Letters · 58

Substituted imidazopyridazines are potent and selective inhibitors of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1)

2013 · Timothy M. Chapman, Simon A. Osborne, et al. · Bioorganic & Medicinal Chemistry Letters · 55

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Imidazopyridazine Inhibitors of Plasmodium falciparum Calcium-Dependent Protein Kinase 1 Also Target Cyclic GMP-Dependent Protein Kinase and Heat Shock Protein 90 To Kill the Parasite at Different Stages of Intracellular Development

2015 · Judith L. Green, Robert W. Moon, et al. · Antimicrobial Agents and Chemotherapy · 53

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Optimization of an Imidazopyridazine Series of Inhibitors of Plasmodium falciparum Calcium-Dependent Protein Kinase 1 (PfCDPK1)

2014 · Timothy M. Chapman, Simon A. Osborne, et al. · Journal of Medicinal Chemistry · 53

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Ligand-Controlled Selectivity in the Desymmetrization of meso Cyclopenten-1,4-diols via Rhodium(I)-Catalyzed Addition of Arylboronic Acids

2010 · Frederic Menard, David Perez, et al. · The Journal of Organic Chemistry · 52

Design, Synthesis, and Testing of Potent, Selective Hepsin Inhibitors via Application of an Automated Closed-Loop Optimization Platform

2018 · Shishir M. Pant, Amanda Mukonoweshuro, et al. · Journal of Medicinal Chemistry · 44

Biochemical and Antiparasitic Properties of Inhibitors of the Plasmodium falciparum Calcium-Dependent Protein Kinase PfCDPK1

2014 · Keith H. Ansell, Hayley M. Jones, et al. · Antimicrobial Agents and Chemotherapy · 34

Catechols and 3-hydroxypyridones as inhibitors of the DNA repair complex ERCC1-XPF

2015 · Timothy M. Chapman, Kevin J. Gillen, et al. · Bioorganic & Medicinal Chemistry Letters · 31

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N-Hydroxyimides and hydroxypyrimidinones as inhibitors of the DNA repair complex ERCC1–XPF

2015 · Timothy M. Chapman, Claire Wallace, et al. · Bioorganic & Medicinal Chemistry Letters · 24

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Synthesis and evaluation of novel cyclopentane urea FPR2 agonists and their potential application in the treatment of cardiovascular inflammation

2021 · Monika Maciuszek, Almudena Ortega-Gomez, et al. · European Journal of Medicinal Chemistry · 14

Design, synthesis, and biological evaluation of novel pyrrolidinone small-molecule Formyl peptide receptor 2 agonists

2021 · Monika Maciuszek, Almudena Ortega-Gomez, et al. · European Journal of Medicinal Chemistry · 6

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Rhodium‐Catalyzed Asymmetric Allylic Substitution with Boronic Acid Nucleophiles.

2007 · Frederic Menard, Timothy M. Chapman, et al. · ChemInform · 2

Discovery of a Selective Lysosomal Alpha-mannosidase Inhibitor From an Imino-sugar Library

2014 · Chang Y-P., M Muckeen, et al. · Journal of Peptide Science

ChemInform Abstract: Ligand‐Controlled Selectivity in the Desymmetrization of meso Cyclopenten‐1,4‐diols via Rhodium(I)‐Catalyzed Addition of Arylboronic Acids.

2010 · Frederic Menard, David Perez, et al. · ChemInform

ChemInform Abstract: Novel Cyclic Sugar Imines: Carbohydrate Mimics and Easily Elaborated Scaffolds for Aza‐Sugars.

2002 · Benjamin G. Davis, Michael A. T. Maughan, et al. · ChemInform

Works count: 20

Citation count: 825

H-index: 14

I10-index: 15