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Daniel Lesieur

New selective ligands of human cloned melatonin MT1 and MT2 receptors
2003 · Valérie Audinot, François Mailliet, et al. · Naunyn-Schmiedeberg s Archives of Pharmacology · 256
Novel naphthalenic ligands with high affinity for the melatonin receptor
1992 · S. Yous, J. Andrieux, et al. · Journal of Medicinal Chemistry · 241
Synthesis and Structure-Activity Relationships of Novel Naphthalenic and Bioisosteric Related Amidic Derivatives as Melatonin Receptor Ligands
1994 · Patrick Depreux, Daniel Lesieur, et al. · Journal of Medicinal Chemistry · 148
Three-Dimensional Quantitative Structure−Activity Relationships of Cyclo-oxygenase-2 (COX-2) Inhibitors: A Comparative Molecular Field Analysis
2001 · Philippe Chavatte, Saïd Yous, et al. · Journal of Medicinal Chemistry · 111
Benzoselenazolinone Derivatives Designed To Be Glutathione Peroxidase Mimetics Feature Inhibition of Cyclooxygenase/5-Lipoxygenase Pathways and Anti-inflammatory Activity
1994 · Vincent Galet, Jean-Luc Bernier, et al. · Journal of Medicinal Chemistry · 107
Synthesis and Structure−Affinity−Activity Relationships of Novel Benzofuran Derivatives as MT2 Melatonin Receptor Selective Ligands
2002 · Valérie Wallez, Sophie Durieux-Poissonnier, et al. · Journal of Medicinal Chemistry · 94
Therapeutic Perspectives for Melatonin Agonists and Antagonists
2003 · P. Delagrange, J. Atkinson, et al. · Journal of Neuroendocrinology · 69
Design and Synthesis of Naphthalenic Dimers as Selective MT1Melatoninergic Ligands
2003 · Carole Descamps-François, Saïd Yous, et al. · Journal of Medicinal Chemistry · 66
Substrate Specificity and Inhibition Studies of Human SerotoninN-Acetyltransferase
2000 · Gilles Ferry, Armelle Loynel, et al. · Journal of Biological Chemistry · 62
Characterisation of human melatonin mt1 and MT2 receptors by CRE-luciferase reporter assay
2000 · Shaun Conway, Sarah J. Canning, et al. · European Journal of Pharmacology · 60
AlCl3-DMF Reagent in the Friedel-Crafts Reaction. Application to the Acylation Reaction of 2(3H)-Benzothiazolones
1994 · Said Yous, Jacques H. Poupaert, et al. · The Journal of Organic Chemistry · 60
Structure-activity relationships in a series of melatonin analogues with the low-density lipoprotein oxidation model
1999 · Andrea Gozzo, Daniel Lesieur, et al. · Free Radical Biology and Medicine · 54
Regioselectivity in the c-acylation of 2(3H)-benzoxazolones
1991 · Hocine Aichaoui, Jacques H. Poupaert, et al. · Tetrahedron · 48
Pictet–Spengler heterocyclizations via microwave-assisted degradation of DMSO
2005 · Christophe Mésangeau, Saïd Yous, et al. · Tetrahedron Letters · 47
Effect of melatonin on motility pattern of small intestine in rats and its inhibition by melatonin receptor antagonist S 22153
2000 · A. Merle, Ph Delagrange, et al. · Journal of Pineal Research · 47
Pharmacophoric Search and 3D-QSAR Comparative Molecular Field Analysis Studies on Agonists of Melatonin Sheep Receptors
1998 · Christophe Marot, Philippe Chavatte, et al. · Journal of Medicinal Chemistry · 47
Effects of both a melatonin agonist and antagonist on seasonal changes in body mass and energy intake in the garden dormouse.
1996 · S Le Gouic, P Delagrange, et al. · PubMed · 47
Pharmacokinetics of Levamisole in healthy subjects and cancer patients
1982 · M. Luyckx, F. Rousseau, et al. · European Journal of Drug Metabolism and Pharmacokinetics · 45
Molecular pharmacology of the ovine melatonin receptor: comparison with recombinant human MT1 and MT2 receptors
2003 · François Mailliet, Valérie Audinot, et al. · Biochemical Pharmacology · 41
A Convenient and efficient method for the preparation of 6‐Acyl‐2(3H)‐benzoxazolones
1992 · Hocine Aichaoui, Daniel Lesieur, et al. · Journal of Heterocyclic Chemistry · 40
Docking Study of Ligands into the Colchicine Binding Site of Tubulin
2004 · Amaury Farce, Cedric Loge, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 39
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Synthesis of Nitroindole Derivatives with High Affinity and Selectivity for Melatoninergic Binding Sites MT3
2002 · Véronique Leclerc, Saïd Yous, et al. · Journal of Medicinal Chemistry · 39
Novel Benzothiazolin-2-one and Benzoxazin-3-one Arylpiperazine Derivatives with Mixed 5HT1A/D2Affinity as Potential Atypical Antipsychotics
1998 · Thierry Taverne, Ousmane Diouf, et al. · Journal of Medicinal Chemistry · 39
S14080, a peripheral analgesic acting by release of an endogenous circulating opioid‐like substance
1995 · Sérgio H. Ferreira, Berenice B. Lorenzetti, et al. · British Journal of Pharmacology · 38
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Synthesis and biological activity of conformationally restricted tricyclic analogs of the hormone melatonin
1996 · V. Leclerc, P. Depreux, et al. · Bioorganic & Medicinal Chemistry Letters · 36
Works count: 173
Citation count: 2,818
H-index: 31
I10-index: 61
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