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Author

Masayuki Matsukura

Observed names: M. MATSUKURA, Masayuki MATSUKURA
Institution: Eisai (Japan)
Observed institution: Eisai (Japan)
OpenAlex ID: A5041422487
Lenvatinib, an angiogenesis inhibitor targeting VEGFR/FGFR, shows broad antitumor activity in human tumor xenograft models associated with microvessel density and pericyte coverage
2014 · Yuji Yamamoto, Junji Matsui, et al. · Vascular Cell · 518
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4-Benzylamino-1-chloro-6-substituted Phthalazines: Synthesis and Inhibitory Activity toward Phosphodiesterase 5
1998 · Nobuhisa Watanabe, Yasuhiro Kabasawa, et al. · Journal of Medicinal Chemistry · 215
In Vitro Activity of E1210, a Novel Antifungal, against Clinically Important Yeasts and Molds
2011 · Mamiko Miyazaki, Takaaki Horii, et al. · Antimicrobial Agents and Chemotherapy · 205
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Efficacy of Oral E1210, a New Broad-Spectrum Antifungal with a Novel Mechanism of Action, in Murine Models of Candidiasis, Aspergillosis, and Fusariosis
2011 · Katsura Hata, Takaaki Horii, et al. · Antimicrobial Agents and Chemotherapy · 156
2-Alkynyl-8-aryl-9-methyladenines as Novel Adenosine Receptor Antagonists: Their Synthesis and Structure−Activity Relationships toward Hepatic Glucose Production Induced via Agonism of the A2BReceptor
2000 · Hitoshi Harada, Osamu Asano, et al. · Journal of Medicinal Chemistry · 113
E7386, a Selective Inhibitor of the Interaction between β-Catenin and CBP, Exerts Antitumor Activity in Tumor Models with Activated Canonical Wnt Signaling
2021 · Kazuhiko Yamada, Yusaku Hori, et al. · Cancer Research · 71
Synthesis and evaluation of novel antifungal agents-quinoline and pyridine amide derivatives
2010 · Kazutaka Nakamoto, Itaru Tsukada, et al. · Bioorganic & Medicinal Chemistry Letters · 47
Synthesis and Antiarrhythmic Activity of 2,2-Dialkyl-1'-(N-substituted aminoalkyl)-spiro-(chroman-4,4'-imidazolidine)-2',5'-diones.
1992 · Masayuki MATSUKURA, Yoshiharu DAIKU, et al. · Chemical and Pharmaceutical Bulletin · 47
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Synthesis of (2R)-1-(4-Chloro-2-pyridyl)-2-(2-pyridyl)ethylamine: A Selective Oxime Reduction and Crystallization-Induced Asymmetric Transformation
1996 · Shigeto Negi, Masayuki Matsukura, et al. · Synthesis · 46
4-(3-Chloro-4-methoxybenzyl)aminophthalazines: Synthesis and Inhibitory Activity toward Phosphodiesterase 5
2000 · Nobuhisa Watanabe, Hideyuki Adachi, et al. · Journal of Medicinal Chemistry · 44
Ten-Gram-Scale Total Synthesis of the Anticancer Drug Candidate E7130 to Supply Clinical Trials
2024 · Yosuke Kaburagi, Kazunobu Kira, et al. · Organic Letters · 15
An Effective Synthesis of a (Pyridin-3-yl)isoxazole via 1,3-Dipolar Cycloaddition Using ZnCl2: Synthesis of a (2-Aminopyridin-3-yl)isoxazole Derivative and Its Antifungal Activity
2010 · Keigo Tanaka, Satoshi Inoue, et al. · Chemistry Letters · 15
What Does It Take to Develop Structurally Complex Molecules by Total Synthesis? Rapid Process Development and GMP Manufacturing of E7130 Drug Substance for First-in-Human Clinical Study
2024 · Takeo Sasaki, Kenzo Yahata, et al. · Organic Process Research & Development · 11
Discovery and development of aryl-fused imidazole-based angiotensin II antagonists
1994 · Kazutoshi Miyake, Masayuki Matsukura, et al. · Bioorganic & Medicinal Chemistry Letters · 7
Abstract 5177: E7386 : First-in-class orally active CBP/beta-catenin modulator as an anticancer agent
2017 · Kazuhiko Yamada, Yusaku Hori, et al. · Cancer Research · 6
Data from E7386, a Selective Inhibitor of the Interaction between β-Catenin and CBP, Exerts Antitumor Activity in Tumor Models with Activated Canonical Wnt Signaling
2023 · Kazuhiko Yamada, Yusaku Hori, et al.
Supplementary Materials and Methods from E7386, a Selective Inhibitor of the Interaction between β-Catenin and CBP, Exerts Antitumor Activity in Tumor Models with Activated Canonical Wnt Signaling
2023 · Kazuhiko Yamada, Yusaku Hori, et al.
Supplementary Table S2 from E7386, a Selective Inhibitor of the Interaction between β-Catenin and CBP, Exerts Antitumor Activity in Tumor Models with Activated Canonical Wnt Signaling
2023 · Kazuhiko Yamada, Yusaku Hori, et al.
Supplementary Table S3 from E7386, a Selective Inhibitor of the Interaction between β-Catenin and CBP, Exerts Antitumor Activity in Tumor Models with Activated Canonical Wnt Signaling
2023 · Kazuhiko Yamada, Yusaku Hori, et al.
Supplementary Tables from E7386, a Selective Inhibitor of the Interaction between β-Catenin and CBP, Exerts Antitumor Activity in Tumor Models with Activated Canonical Wnt Signaling
2023 · Kazuhiko Yamada, Yusaku Hori, et al.
Supplementary Figures from E7386, a Selective Inhibitor of the Interaction between β-Catenin and CBP, Exerts Antitumor Activity in Tumor Models with Activated Canonical Wnt Signaling
2023 · Kazuhiko Yamada, Yusaku Hori, et al.
ChemInform Abstract: 4‐Benzylamino‐1‐chloro‐6‐Substituted Phthalazines: Synthesis and Inhibitory Activity Toward Phosphodiesterase 5.
1998 · N. WATANABE, Y. KABASAWA, et al. · ChemInform
ChemInform Abstract: Synthesis of (2R)‐1‐(4‐Chloro‐2‐pyridyl)‐2‐(2‐pyridyl)ethylamine: A Selective Oxime Reduction and Crystallization‐Induced Asymmetric Transformation.
1996 · S. NEGI, M. MATSUKURA, et al. · ChemInform
ChemInform Abstract: Discovery and Development of Aryl‐Fused Imidazole‐Based Angiotensin II Antagonists
1994 · K. MIYAKE, M. MATSUKURA, et al. · ChemInform
ChemInform Abstract: Synthesis and Cardiovascular Activity of Phenylalkylamine Derivatives. Part 1. Potential Specific Bradycardic Agents.
1993 · F. OZAKI, M. MATSUKURA, et al. · ChemInform
Works count: 25
Citation count: 1,516
H-index: 12
I10-index: 13
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