Author

Harry Cheung

Institutions: Novartis (Switzerland), Novartis (United States)

Observed institutions: Novartis (Switzerland), Novartis (United States), Elan Pharmaceuticals, Inc. (Ireland)

OpenAlex ID: A5044044762

Design and Synthesis of Tri-Ring P3 Benzamide-Containing Aminonitriles as Potent, Selective, Orally Effective Inhibitors of Cathepsin K

2005 · James T. Palmer, Clifford Bryant, et al. · Journal of Medicinal Chemistry · 95

Keto-1,3,4-oxadiazoles as cathepsin K inhibitors

2006 · James T. Palmer, Bernard L. Hirschbein, et al. · Bioorganic & Medicinal Chemistry Letters · 73

Peptide Ketobenzoxazole Inhibitors Bound to Cathepsin K

2003 · Mary E. McGrath, Paul A. Sprengeler, et al. · Biochemistry · 41

3,4-Disubstituted azetidinones as selective inhibitors of the cysteine protease cathepsin K. Exploring P3 elements for potency and selectivity

2005 · Eduardo L. Setti, Dana Davis, et al. · Bioorganic & Medicinal Chemistry Letters · 29

Design and synthesis of tetracyclic nonpeptidic biaryl nitrile inhibitors of cathepsin K

2006 · Eduardo L. Setti, Shankar Venkatraman, et al. · Bioorganic & Medicinal Chemistry Letters · 9

Development of a Novel β-Secretase Binding Assay Using the AlphaScreen Platform

2013 · Zhao Ren, Danny Tam, et al. · SLAS DISCOVERY · 7

Discovery of IID432 for Chagas Disease: A Cyanotriazole Inhibitor of Trypanosoma cruzi Topoisomerase II Achieves Sterile Cure After Short-Term Treatment in a Chronic Infection Model

2026 · Olivier René, Manuel Saldivia, et al. · Journal of Medicinal Chemistry · 2

Keto‐1,3,4‐oxadiazoles as Cathepsin K Inhibitors.

2006 · James T. Palmer, Bernard L. Hirschbein, et al. · ChemInform · 1

Discovery of a Pyrazine-2-Carboxamide Derivative as a Potent Plasmodium falciparum Inhibitor with Potential for Single-Dose Cure

2026 · Vanessa M. Marx, Anne-Catherine Mata, et al. · Journal of Medicinal Chemistry

Design and Synthesis of Tetracyclic Nonpeptidic Biaryl Nitrile Inhibitors of Cathepsin K.

2006 · Eduardo L. Setti, Shankar Venkatraman, et al. · ChemInform

3,4‐Disubstituted Azetidinones as Selective Inhibitors of the Cysteine Protease Cathepsin K. Exploring P3 Elements for Potency and Selectivity.

2005 · Eduardo L. Setti, Dana Davis, et al. · ChemInform

Works count: 11

Citation count: 257

H-index: 6

I10-index: 4