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Yves Mérand

Observed names: Y Merand, Y Mérand, Y. MERAND, Y. Merand, Y. Mérand, YVES MÉRAND, Yves Merand
OpenAlex ID: A5047828126
EM-652 (SCH 57068), a third generation SERM acting as pure antiestrogen in the mammary gland and endometrium
1999 · Fernand Labrie, Claude Labrie, et al. · The Journal of Steroid Biochemistry and Molecular Biology · 161
(S)-(+)-4-[7-(2,2-Dimethyl-1-oxopro- poxy)-4-methyl-2-[4-[2-(1-piperidinyl)- ethoxy]phenyl]-2H-1-benzopyran-3-yl]- phenyl 2,2-Dimethylpropanoate (EM-800): A Highly Potent, Specific, and Orally Active Nonsteroidal Antiestrogen
1997 · Sylvain Gauthier, Brigitte Caron, et al. · Journal of Medicinal Chemistry · 156
Regulation of Progesterone-Binding Breast Cyst Protein GCDFP-24 Secretion by Estrogens and Androgens in Human Breast Cancer Cells: A New Marker of Steroid Action in Breast Cancer*
1990 · JACQUES SIMARD, SOPHIE DAUVOIS, et al. · Endocrinology · 110
Age-related changes in central nervous system enkephalins and substance P
1981 · A. Dupont, P. Savard, et al. · Life Sciences · 96
Changes in the β-endorphin content of discrete hypothalamic nuclei during the estrous cycle of the rat
1981 · Nicholas Barden, Yves Mérand, et al. · Brain Research · 90
Antiestrogenic properties of keoxifene,trans-4-hydroxytamoxifen, and ICI 164384, a new steroidal antiestrogen, in ZR-75-1 human breast cancer cells
1989 · Richard Poulin, Yves Merand, et al. · Breast Cancer Research and Treatment · 86
beta-Endorphin and met-enkephalins: their distribution, modulation by estrogens and haloperidol, and role in neuroendocrine control.
1980 · A Dupont, N Barden, et al. · PubMed · 82
Synthesis and biological activity of new halo-steroidal antiestrogens
1991 · Charles Levesque, Yves Merand, et al. · Journal of Medicinal Chemistry · 81
Characterization of the effects of the novel non-steroidal antiestrogen EM-800 on basal and estrogen-induced proliferation of T-47D, ZR-75-1 and MCF-7 human breast cancer cellsin vitro
1997 · Jacques Simard, Claude Labrie, et al. · International Journal of Cancer · 74
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Novel compounds inhibit estrogen formation and action.
1992 · C Labrie, C Martel, et al. · PubMed · 73
Blockade of the stimulatory effect of estrogens, OH-tamoxifen, OH-toremifene, droloxifene, and raloxifene on alkaline phosphatase activity by the antiestrogen EM-800 in human endometrial adenocarcinoma Ishikawa cells.
1997 · J Simard, R Sanchez, et al. · PubMed · 70
Additive inhibitory effects of an androgen and the antiestrogen EM-170 on estradiol-stimulated growth of human ZR-75-1 breast tumors in athymic mice.
1991 · S Dauvois, C S Geng, et al. · PubMed · 69
Regional distributions of somatostatin and cholecystokinin-like immunoreactivities in rat and bovine brain
1981 · Nicholas Barden, Yves Mérand, et al. · Peptides · 67
Differential distribution of β-endorphin and enkephalins in rat and bovine brain
1980 · André Dupont, Jérôme Lépine, et al. · Regulatory Peptides · 61
Comparative effects of 28-day treatment with the new anti-estrogen EM-800 and tamoxifen on estrogen-sensitive parameters in intact mice
1997 · Shouqi Luo, Céline Martel, et al. · International Journal of Cancer · 53
Binding characteristics of novel nonsteroidal antiestrogens to the rat uterine estrogen receptors
1998 · Céline Martel, Louis Provencher, et al. · The Journal of Steroid Biochemistry and Molecular Biology · 44
Enzymic inactivation of neurotensin by hypothalamic and brain extracts of the rat
1978 · A. Dupont, Y. Mérand · Life Sciences · 44
Effect of Neonatal Thyroid Deficiency on the Catecholamine, Substance P, and Thyrotropin-Releasing Hormone Contents of Discrete Rat Brain Nuclei
1981 · ANDRÉ DUPONT, JEAN-H. DUSSAULT, et al. · Endocrinology · 40
Effect of neonatal hypothyroidism on the serotonin system of the rat brain
1984 · Pierre Savard, Yves Mérand, et al. · Brain Research · 38
Effects of thyroid state on serotonin, 5-hydroxyindoleacetic acid and substance P contents in discrete brain nuclei of adult rats
1983 · P. Savard, Y. Mérand, et al. · Neuroscience · 38
Comparison of the Effects of the New Orally Active Antiestrogen EM-800 with ICI 182 780 and Toremifene on Estrogen-Sensitive Parameters in the Ovariectomized Mouse
1998 · Céline Martel, Claude Labrie, et al. · Endocrinology · 35
Synthesis and Antiestrogenic Activity of Diaryl Thioether Derivatives
1994 · Donald Poirier, Serge Auger, et al. · Journal of Medicinal Chemistry · 35
Effect of Twenty-Four-Week Treatment with the Antiestrogen EM-800 on Estrogen-Sensitive Parameters in Intact and Ovariectomized Mice
1998 · Shouqi Luo, Antigone Sourla, et al. · Endocrinology · 33
Interactions between Estrogens, Androgens, Progestins, and Glucocorticoids in ZR‐75‐1 Human Breast Cancer Cells
1990 · Fernand Labrie, Richard Poulin, et al. · Annals of the New York Academy of Sciences · 30
Extensive Esterification of Adrenal C19-Δ5-Sex Steroids to Long-Chain Fatty Acids in the ZR-75-1 Human Breast Cancer Cell Line
1989 · R Poulin, D Poirier, et al. · Journal of Biological Chemistry · 30
Works count: 59
Citation count: 2,026
H-index: 25
I10-index: 43
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