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Shigetoshi Kikuchi

Optical Resolution of 2-Amino-1,2-diphenylethanol by Preferential Crystallization and Its Utilization in Fractional Crystallization and Enantioselective Reduction of Prochiral Ketones
1982 · Kazuhiko Saigo, Shigeo Ogawa, et al. · Bulletin of the Chemical Society of Japan · 66
Total Synthesis of Brevenal
2009 · Hiroyoshi Takamura, Shigetoshi Kikuchi, et al. · Organic Letters · 65
Structure-based drug design of 1,3,5-triazine and pyrimidine derivatives as novel FGFR3 inhibitors with high selectivity over VEGFR2
2020 · Ikumi Kuriwaki, Minoru Kameda, et al. · Bioorganic & Medicinal Chemistry · 41
Design and synthesis of novel benzimidazole derivatives as phosphodiesterase 10A inhibitors with reduced CYP1A2 inhibition
2013 · Wataru Hamaguchi, Naoyuki Masuda, et al. · Bioorganic & Medicinal Chemistry · 33
Synthesis, SAR study, and biological evaluation of novel quinoline derivatives as phosphodiesterase 10A inhibitors with reduced CYP3A4 inhibition
2014 · Wataru Hamaguchi, Naoyuki Masuda, et al. · Bioorganic & Medicinal Chemistry · 22
Total synthesis of brevenal
2010 · Hiroyoshi Takamura, Yuji Yamagami, et al. · Tetrahedron · 21
Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency
2021 · Ikumi Kuriwaki, Minoru Kameda, et al. · Bioorganic & Medicinal Chemistry · 16
Solvent-Controlled Stereoselective Formation of a Cyclic Ether in the Lewis Acid-Mediated Allylation of an α-Chloroacetoxy Acyclic Ether. Very High Stereoselectivity in CH3CN vs Low Stereoselectivity in CH2Cl2
2007 · Ilya D. Gridnev, Shigetoshi Kikuchi, et al. · The Journal of Organic Chemistry · 14
Discovery of ASP5878: Synthesis and structure–activity relationships of pyrimidine derivatives as pan-FGFRs inhibitors with improved metabolic stability and suppressed hERG channel inhibitory activity
2022 · Ikumi Kuriwaki, Minoru Kameda, et al. · Bioorganic & Medicinal Chemistry · 11
Addressing phototoxicity observed in a novel series of biaryl derivatives: Discovery of potent, selective and orally active phosphodiesterase 10A inhibitor ASP9436
2015 · Wataru Hamaguchi, Naoyuki Masuda, et al. · Bioorganic & Medicinal Chemistry · 11
Convergent synthesis of the F–K ring segment of brevetoxin B
2003 · Isao Kadota, Naoko Nishina, et al. · Tetrahedron Letters · 6
Near-Infrared Fluorescent Silica Nanoparticles Based on Gold–Silver Alloy Nanoclusters for Clinical Diagnosis
2024 · Hiroaki Ichimaru, Shigetoshi Kikuchi · Chemical and Pharmaceutical Bulletin · 1
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Magnetic Polystyrene Nanoparticles Prepared by Emulsion Solvent-Evaporation for the Chemiluminescent Immunoassay
2024 · Hiroaki Ichimaru, Masashi Kurimoto, et al. · Chemical and Pharmaceutical Bulletin
Preparation of Hydrophobic Bovine-Serum-Albumin-capped Gold Nanoclusters and Encapsulation in Polystyrene Nanoparticles
2024 · Hiroaki Ichimaru, Natsumi Hanazawa, et al. · e-Journal of Surface Science and Nanotechnology
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ChemInform Abstract: Total Synthesis of Brevenal.
2010 · Hiroyoshi Takamura, Yuji Yamagami, et al. · ChemInform
Works count: 15
Citation count: 307
H-index: 10
I10-index: 10
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