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Antony A. Okumu

Observed names: Antony Akura Okumu, Antony Okumu
ORCID: 0000-0002-4641-7843
Observed ORCID: 0000-0002-4641-7843
OpenAlex ID: A5059632504
Optimization of TopoIV Potency, ADMET Properties, and hERG Inhibition of 5-Amino-1,3-dioxane-Linked Novel Bacterial Topoisomerase Inhibitors: Identification of a Lead with In Vivo Efficacy against MRSA
2021 · Yanran Lu, Sandip Vibhute, et al. · Journal of Medicinal Chemistry · 40
1,3-Dioxane-Linked Bacterial Topoisomerase Inhibitors with Enhanced Antibacterial Activity and Reduced hERG Inhibition
2019 · Linsen Li, Antony A. Okumu, et al. · ACS Infectious Diseases · 38
Stereochemical Definition of the Natural Product (6R,10R,13R, 14R,16R,17R,19S,20S,21R,24S,25S,28S,30S,32R,33R,34R,36S,37S,39R)‐Azaspiracid‐3 by Total Synthesis and Comparative Analyses
2017 · Nathaniel T. Kenton, Daniel Adu‐Ampratwum, et al. · Angewandte Chemie International Edition · 24
Synthesis and anti-staphylococcal activity of novel bacterial topoisomerase inhibitors with a 5-amino-1,3-dioxane linker moiety
2018 · Linsen Li, Antony Okumu, et al. · Bioorganic & Medicinal Chemistry Letters · 21
Synthesis of the C22–C40 Domain of the Azaspiracids
2016 · Zhigao Zhang, Yong Chen, et al. · Organic Letters · 16
Novel bacterial topoisomerase inhibitors derived from isomannide
2020 · Antony Okumu, Yanran Lu, et al. · European Journal of Medicinal Chemistry · 15
Total Synthesis of (6R,10R,13R,14R,16R,17R,19S,20R,21R,24S, 25S,28S,30S,32R,33R,34R,36S,37S,39R)‐Azaspiracid‐3 Reveals Non‐Identity with the Natural Product
2017 · Nathaniel T. Kenton, Daniel Adu‐Ampratwum, et al. · Angewandte Chemie International Edition · 13
Stereochemical Definition of the Natural Product (6R,10R,13R, 14R,16R,17R,19S,20S,21R,24S,25S,28S,30S,32R,33R,34R,36S,37S,39R)‐Azaspiracid‐3 by Total Synthesis and Comparative Analyses
2017 · Nathaniel T. Kenton, Daniel Adu‐Ampratwum, et al. · Angewandte Chemie · 5
Total Synthesis of (6R,10R,13R,14R,16R,17R,19S,20R,21R,24S, 25S,28S,30S,32R,33R,34R,36S,37S,39R)‐Azaspiracid‐3 Reveals Non‐Identity with the Natural Product
2017 · Nathaniel T. Kenton, Daniel Adu‐Ampratwum, et al. · Angewandte Chemie · 4
Synthesis of the C1–C19 Domain of Azaspiracid-34
2019 · Antony A. Okumu, Craig J. Forsyth · Organic Letters · 1
Toward Total Synthesis of Azaspiracid-3 and Azaspiracid-34
2016 · Antony A. Okumu · OhioLink ETD Center (Ohio Library and Information Network)
Development of a Safe and Efficient Alkyl Azide Synthesis using Arylsulfonyl Azide
2010 · Antony A. Okumu · OhioLink ETD Center (Ohio Library and Information Network)
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Works count: 12
Citation count: 177
H-index: 7
I10-index: 7
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