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Jörge Beleta

U-BIOPRED clinical adult asthma clusters linked to a subset of sputum omics
2016 · Diane Lefaudeux, Bertrand De Meulder, et al. · Journal of Allergy and Clinical Immunology · 301
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Characterization of Aclidinium Bromide, a Novel Inhaled Muscarinic Antagonist, with Long Duration of Action and a Favorable Pharmacological Profile
2009 · Amadeu Gavaldà, Montserrat Miralpeix, et al. · Journal of Pharmacology and Experimental Therapeutics · 129
IL-17–high asthma with features of a psoriasis immunophenotype
2019 · Jörgen Östling, Marleen van Geest, et al. · Journal of Allergy and Clinical Immunology · 125
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Investigation into the role of phosphodiesterase IV in bronchorelaxation, including studies with human bronchus
1993 · J. Cortijo, J. Bou, et al. · British Journal of Pharmacology · 113
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The human area postrema and other nuclei related to the emetic reflex express cAMP phosphodiesterases 4B and 4D
2010 · F. Mori, S. Pérez-Torres, et al. · Journal of Chemical Neuroanatomy · 90
Adenosine Inhibits Macrophage Colony-Stimulating Factor-Dependent Proliferation of Macrophages Through the Induction of p27 kip-1 Expression
1999 · Jordi Xaus, Annabel F Valledor, et al. · The Journal of Immunology · 84
Pharmacological blockade of CCR1 ameliorates murine arthritis and alters cytokine networksin vivo
2006 · M Amat, C F Benjamim, et al. · British Journal of Pharmacology · 81
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Discovery of Novel Quaternary Ammonium Derivatives of (3R)-Quinuclidinol Esters as Potent and Long-Acting Muscarinic Antagonists with Potential for Minimal Systemic Exposure after Inhaled Administration: Identification of (3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane Bromide (Aclidinium Bromide)
2009 · María Prat, Dolors Fernández, et al. · Journal of Medicinal Chemistry · 73
Characterization of human serotonin 1D and 1B receptors using [ 3H]-GR-125743, a novel radiolabelled serotonin 5HT1D/1B receptor antagonist
1997 · T. Doménech, J. Beleta, et al. · Naunyn-Schmiedeberg s Archives of Pharmacology · 73
Novel Heterocyclic-Fused Pyridazinones as Potent and Selective Phosphodiesterase IV Inhibitors
1997 · Vittorio Dal Piaz, Maria Paola Giovannoni, et al. · Journal of Medicinal Chemistry · 73
Benzyl Derivatives of 2,1,3-Benzo- and Benzothieno[3,2-a]thiadiazine 2,2-Dioxides: First Phosphodiesterase 7 Inhibitors
2000 · Ana Martínez, Ana Castro, et al. · Journal of Medicinal Chemistry · 72
Identification and characterization of serotonin 5-HT4 receptor binding sites in human brain: comparison with other mammalian species
1994 · T. Doménech, J. Beleta, et al. · Molecular Brain Research · 72
Aclidinium bromide, a new, long-acting, inhaled muscarinic antagonist: In vitro plasma inactivation and pharmacological activity of its main metabolites
2010 · Sonia Sentellas, Israel Ramos, et al. · European Journal of Pharmaceutical Sciences · 71
Bronchodilator and anti‐inflammatory activities of glaucine: In vitro studies in human airway smooth muscle and polymorphonuclear leukocytes
1999 · J Cortijo, V Villagrasa, et al. · British Journal of Pharmacology · 69
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Phosphodiesterase inhibitory properties of losartan. design and synthesis of new lead compounds
1998 · Victor Segarra, M. Isabel Crespo, et al. · Bioorganic & Medicinal Chemistry Letters · 59
Characterization of 5‐HT receptors on human pulmonary artery and vein: functional and binding studies
1997 · Julio Cortijo, Miguel Martí‐Cabrera, et al. · British Journal of Pharmacology · 57
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Pharmacological Characterization of Abediterol, a Novel Inhaled β2-Adrenoceptor Agonist with Long Duration of Action and a Favorable Safety Profile in Preclinical Models
2012 · Mònica Aparici, Mireia Gómez-Angelats, et al. · Journal of Pharmacology and Experimental Therapeutics · 53
The in vitro and in vivo profile of aclidinium bromide in comparison with glycopyrronium bromide
2014 · Amadeu Gavaldà, Israel Ramos, et al. · Pulmonary Pharmacology & Therapeutics · 48
Functional and biochemical evidence for diazepam as a cyclic nucleotide phosphodiesterase type 4 inhibitor
1998 · M Carmen Collado, Jorge Beleta, et al. · British Journal of Pharmacology · 40
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Pharmacological characterization of almotriptan: an indolic 5-HT receptor agonist for the treatment of migraine
2000 · Josep Bou, Teresa Domènech, et al. · European Journal of Pharmacology · 36
Inhibition of eotaxin‐mediated human eosinophil activation and migration by the selective cyclic nucleotide phosphodiesterase type 4 inhibitor rolipram
1997 · Luis F Santamaria, Jose Maria Palacios, et al. · British Journal of Pharmacology · 35
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Synthesis and Biological Activity of Pyrido[3′,2′:4,5]thieno[3,2-d]pyrimidines as Phosphodiesterase Type 4 Inhibitors
2010 · Joan Taltavull, Jordi Serrat, et al. · Journal of Medicinal Chemistry · 33
Discovery and Characterization of 4‘-(2-Furyl)-N-pyridin-3-yl-4,5‘-bipyrimidin-2‘-amine (LAS38096), a Potent, Selective, and Efficacious A2BAdenosine Receptor Antagonist
2007 · Bernat Vidal, Arsenio Nueda, et al. · Journal of Medicinal Chemistry · 33
Anticholinergic effects of desloratadine, the major metabolite of loratadine, in rabbit and guinea-pig iris smooth muscle
1999 · Ignasi Cardelús, Francisca Antón, et al. · European Journal of Pharmacology · 30
Heterocyclic-fused 3(2H)-pyridazinones as potent and selective PDE IV inhibitors: Further structure-activity relationships and molecular modelling studies
1998 · Vittorio Dal Piaz, Maria Paola Giovannoni, et al. · European Journal of Medicinal Chemistry · 29
Works count: 73
Citation count: 2,208
H-index: 27
I10-index: 36
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