Author

Sándor Kolok

Observed names: S KOLOK, S Kolok, S. Kolok, Sandor Kolok

Observed institutions: Gedeon Richter (Hungary), Budapest University of Technology and Economics

OpenAlex ID: A5066254271

Tolperisone-Type Drugs Inhibit Spinal Reflexes via Blockade of Voltage-Gated Sodium and Calcium Channels

2005 · Pál Kocsis, Sándor Farkas, et al. · Journal of Pharmacology and Experimental Therapeutics · 66

NR2B subunit selective NMDA antagonists inhibit neurotoxic effect of alcohol-withdrawal in primary cultures of rat cortical neurones

2003 · J Nagy, Csilla Horváth, et al. · Neurochemistry International · 60

Differential alterations in the expression of NMDA receptor subunits following chronic ethanol treatment in primary cultures of rat cortical and hippocampal neurones

2002 · József Nagy, Sándor Kolok, et al. · Neurochemistry International · 52

Selective NR1/2BN-Methyl- d -aspartate Receptor Antagonists among Indole-2-carboxamides and Benzimidazole-2-carboxamides

2007 · István Borza, Éva Bozó, et al. · Journal of Medicinal Chemistry · 45

Oxamides as novel NR2B selective NMDA receptor antagonists

2004 · Gizella Barta-Szalai, István Borza, et al. · Bioorganic & Medicinal Chemistry Letters · 45

Kynurenic acid amides as novel NR2B selective NMDA receptor antagonists

2006 · István Borza, Sándor Kolok, et al. · Bioorganic & Medicinal Chemistry Letters · 39

Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists

2003 · István Borza, Sándor Kolok, et al. · Bioorganic & Medicinal Chemistry Letters · 37

Role of Altered Structure and Function of NMDA Receptors in Development of Alcohol Dependence

2005 · J. Nagy, S. Kolok, et al. · Current Neuropharmacology · 32

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Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications

2017 · János Galambos, Attila Bielik, et al. · Journal of Medicinal Chemistry · 30

Quinolinyl- and phenantridinyl-acetamides as bradykinin B1 receptor antagonists

2012 · János Éles, Gyula Beke, et al. · Bioorganic & Medicinal Chemistry Letters · 26

4-Aryl-3-arylsulfonyl-quinolines as negative allosteric modulators of metabotropic GluR5 receptors: From HTS hit to development candidate

2016 · János Galambos, György Domány, et al. · Bioorganic & Medicinal Chemistry Letters · 22

Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists

2010 · János Galambos, Gábor Wágner, et al. · Bioorganic & Medicinal Chemistry Letters · 22

Benzimidazole-2-carboxamides as novel NR2B selective NMDA receptor antagonists

2006 · István Borza, Sándor Kolok, et al. · Bioorganic & Medicinal Chemistry Letters · 22

Inducible expression and pharmacology of recombinant NMDA receptors, composed of rat NR1a/NR2B subunits

2003 · József Nagy, András Boros, et al. · Neurochemistry International · 22

Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs

2010 · Gábor Wágner, Csaba Wéber, et al. · Bioorganic & Medicinal Chemistry Letters · 20

Indole-2-carboxamidines as novel NR2B selective NMDA receptor antagonists

2005 · István Borza, Sándor Kolok, et al. · Bioorganic & Medicinal Chemistry Letters · 19

Discovery of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor: Scaffold hopping approach

2021 · István Ledneczki, Pál Tapolcsányi, et al. · European Journal of Medicinal Chemistry · 17

Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Lead optimization

2015 · Katalin Nógrádi, Gábor Wágner, et al. · Bioorganic & Medicinal Chemistry Letters · 16

Fragment Based Optimization of Metabotropic Glutamate Receptor 2 (mGluR2) Positive Allosteric Modulators in the Absence of Structural Information

2018 · György Szabó, György I. Túrós, et al. · Journal of Medicinal Chemistry · 14

Analysis of functional selectivity through G protein-dependent and -independent signaling pathways at the adrenergic α2C receptor

2014 · Dalma Kurko, Zoltán Kapui, et al. · Brain Research Bulletin · 13

Inducible expression and pharmacological characterization of recombinant rat NR1a/NR2A NMDA receptors

2005 · Dalma Kurkó, Péter Dezső, et al. · Neurochemistry International · 13

Cell-based and virtual fragment screening for adrenergic α2C receptor agonists

2015 · Edit Szőllősi, Amrita Bobok, et al. · Bioorganic & Medicinal Chemistry · 12

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Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Hit-to-lead optimization

2014 · Katalin Nógrádi, Gábor Wágner, et al. · Bioorganic & Medicinal Chemistry Letters · 11

Functional characterization of sodium channel blockers by membrane potential measurements in cerebellar neurons: Prediction of compound preference for the open/inactivated state

2006 · S KOLOK, J NAGY, et al. · Neurochemistry International · 11

Comparative pharmacology of adrenergic α2C receptors coupled to Ca2+ signaling through different Gα proteins

2009 · Dalma Kurko, Zsófia Bekes, et al. · Neurochemistry International · 9

Works count: 39

Citation count: 708

H-index: 17

I10-index: 24