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Cristina Gardelli

Observed names: C. GARDELLI, C. Gardelli, Gardelli Cristina, Gardelli, Cristina
ORCID: 0000-0003-1169-2180
Observed ORCID: 0000-0003-1169-2180
OpenAlex ID: A5073858751
Discovery of Raltegravir, a Potent, Selective Orally Bioavailable HIV-Integrase Inhibitor for the Treatment of HIV-AIDS Infection
2008 · Vincenzo Summa, Alessia Petrocchi, et al. · Journal of Medicinal Chemistry · 652
4,5-Dihydroxypyrimidine Carboxamides and N-Alkyl-5-hydroxypyrimidinone Carboxamides Are Potent, Selective HIV Integrase Inhibitors with Good Pharmacokinetic Profiles in Preclinical Species
2006 · Vincenzo Summa, Alessia Petrocchi, et al. · Journal of Medicinal Chemistry · 104
Enantioselective Total Synthesis of the Antitumor Macrolide Rhizoxin D
2003 · Jennifer A. Lafontaine, David P. Provencal, et al. · The Journal of Organic Chemistry · 92
Regiochemical control of the ring opening of 1,2-epoxides by means of chelating processes. 5. Synthesis and reactions of some 2,3-epoxy-1-alkanol derivatives
1993 · Marco Chini, Paolo Crotti, et al. · The Journal of Organic Chemistry · 89
Dihydroxypyrimidine-4-carboxamides as Novel Potent and Selective HIV Integrase Inhibitors
2007 · Paola Pace, M. Emilia Di Francesco, et al. · Journal of Medicinal Chemistry · 80
Discovery and Synthesis of HIV Integrase Inhibitors: Development of Potent and Orally Bioavailable N-Methyl Pyrimidones
2007 · Cristina Gardelli, Emanuela Nizi, et al. · Journal of Medicinal Chemistry · 67
Regio- and Stereoselective Synthesis of β-Halohydrins from 1,2-Epoxides with Ammonium Halides in the Presence of Metal Salts
1992 · Marco Chini, Paolo Crotti, et al. · Tetrahedron · 59
Phosphoramidate Prodrugs of 2′-C-Methylcytidine for Therapy of Hepatitis C Virus Infection
2009 · Cristina Gardelli, Barbara Attenni, et al. · Journal of Medicinal Chemistry · 55
Design and Synthesis of Bicyclic Pyrimidinones as Potent and Orally Bioavailable HIV-1 Integrase Inhibitors
2008 · Ester Muraglia, Olaf Kinzel, et al. · Journal of Medicinal Chemistry · 53
Regiochemical control of the ring opening of 1,2-epoxides by means of chelating processes. 8. Synthesis and ring opening reactions of cis- and trans- oxides derived from 3-benzyloxycyclohexene and 2-benzyloxy-5,6-dihydro-2H-pyran
1994 · Federico Calvani, Paolo Crotti, et al. · Tetrahedron · 52
Discovery of Highly Isoform Selective Orally Bioavailable Phosphoinositide 3-Kinase (PI3K)-γ Inhibitors
2018 · Nils Pemberton, Mickael Mogemark, et al. · Journal of Medicinal Chemistry · 45
The Design and Enzyme-Bound Crystal Structure of Indoline Based Peptidomimetic Inhibitors of Hepatitis C Virus NS3 Protease
2004 · Jesus M. Ontoria, Stefania Di Marco, et al. · Journal of Medicinal Chemistry · 42
Metal Salt-Promoted Alcoholysis of 1,2-Epoxides
1992 · Marco Chini, Paolo Crotti, et al. · Synlett · 36
The enantioselective total synthesis of the antitumor macrolide natural product rhizoxin D
1999 · Jennifer A. Lafontaine, David P. Provencal, et al. · Tetrahedron Letters · 33
Synthesis and evaluation of novel phosphoramidate prodrugs of 2′-methyl cytidine as inhibitors of hepatitis c virus NS5B polymerase
2009 · Monica Donghi, Barbara Attenni, et al. · Bioorganic & Medicinal Chemistry Letters · 32
Rhizoxin synthetic studies. 2. Synthesis of the left hand [C(10) to C(19)] and polyene fragments
1995 · David P. Provencal, Cristina Gardelli, et al. · Tetrahedron Letters · 32
Regiochemical Control of the Ring Opening of 1,2-Epoxides by Means of Chelating Processes. 7. Synthesis and Ring-Opening Reactions of cis- and trans-Oxides Derived from 2-(Benzyloxy)-3,6-dihydro-2H-pyran
1994 · Marco Chini, Paolo Crotti, et al. · The Journal of Organic Chemistry · 32
Cyclic phosphoramidates as prodrugs of 2′-C-methylcytidine
2009 · Malte Meppen, Barbara Pacini, et al. · European Journal of Medicinal Chemistry · 31
Regiochemical control of the ring opening of 1,2-epoxides by means of chelating processes. 4. Synthesis and reactions of the cis- and trans-oxides derived from 3-[(benzyloxy)methyl]cyclohexene
1992 · Marco Chini, Paolo Crotti, et al. · The Journal of Organic Chemistry · 31
Regiochemical control of the ring opening of 1:2-epoxides by means of chelating processes. 10. Synthesis and ring opening reactions of mono- and difunctionalized cis and trans aliphatic oxirane systems
1995 · Francesca Azzena, Federico Calvani, et al. · Tetrahedron · 30
Regiochemical Control of the Ring Opening of Aziridines by Means of Chelating Processes. Synthesis and Ring-Opening Reactions of cis- and trans-Aziridines Derived from 4-(Benzyloxy)cyclohexene
1995 · Paolo Crotti, Lucilla Favero, et al. · The Journal of Organic Chemistry · 27
Regiochemical control of the ring opening of 1,2-epoxides by means of chelating processes. 6. Opening reactions of 3,4-epoxytetrahydropyran
1994 · Chini Marco, Crotti Paolo, et al. · Tetrahedron · 25
Identification and Optimization of Pyrrolidine Derivatives as Highly Potent Ghrelin Receptor Full Agonists
2020 · Martin Cooper, Antonio Llinas, et al. · Journal of Medicinal Chemistry · 24
Macrophage Activation Status Rather than Repolarization Is Associated with Enhanced Checkpoint Activity in Combination with PI3Kγ Inhibition
2021 · Larissa S. Carnevalli, Molly A. Taylor, et al. · Molecular Cancer Therapeutics · 21
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Synthesis of a hexahydropyrimido[1,2-a]azepine-2-carboxamide derivative useful as an HIV integrase inhibitor
2007 · Marco Ferrara, Benedetta Crescenzi, et al. · Tetrahedron Letters · 20
Works count: 77
Citation count: 1,913
H-index: 23
I10-index: 33
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