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Johannes Brussee

Preparation and NMR characterization of highly substitutedN-trimethyl chitosan chloride
1998 · A.B. Sieval, M. Thanou, et al. · Carbohydrate Polymers · 437
On the mechanism of the formation of s(−)-(1, 1'-binaphthalene)-2,2'-diol via copper(II)amine complexes
1985 · J. Brussee, J.L.G. Groenendijk, et al. · Tetrahedron · 196
Chiral Induction Effects in Ruthenium(II) Amino Alcohol Catalysed Asymmetric Transfer Hydrogenation of Ketones: An Experimental and Theoretical Approach
2000 · Daniëlle G. I. Petra, Joost N. H. Reek, et al. · Chemistry - A European Journal · 164
New, Non-Adenosine, High-Potency Agonists for the Human Adenosine A2B Receptor with an Improved Selectivity Profile Compared to the Reference Agonist N-Ethylcarboxamidoadenosine
2004 · Margot W. Beukers, Lisa C. W. Chang, et al. · Journal of Medicinal Chemistry · 154
2-Amino-6-furan-2-yl-4-substituted Nicotinonitriles as A2A Adenosine Receptor Antagonists
2008 · Monica Mantri, Olivier de Graaf, et al. · Journal of Medicinal Chemistry · 151
Thermodynamic and structural aspects of the skin barrier
1991 · J.A. Bouwstra, M.A. de Vries, et al. · Journal of Controlled Release · 130
Pyrazole Derivatives as Partial Agonists for the Nicotinic Acid Receptor
2003 · T. van Herk, J. Brussee, et al. · Journal of Medicinal Chemistry · 116
A highly stereoselective synthesis of s(-)-[1,1′-binaphthalene]-2,2′-diol
1983 · J. Brussee, A.C.A. Jansen · Tetrahedron Letters · 114
A Series of Ligands Displaying a Remarkable Agonistic−Antagonistic Profile at the Adenosine A1 Receptor
2004 · Lisa C. W. Chang, Jacobien K. von Frijtag Drabbe Künzel, et al. · Journal of Medicinal Chemistry · 113
Bio-organic synthesis of optically active cyanohydrins and acyloins
1988 · J. Brussee, E.C. Roos, et al. · Tetrahedron Letters · 111
Synthesis of Optically Active Cyanohydrins Using Almond Meal
1991 · P. Zandbergen, J. van der Linden, et al. · Synthetic Communications · 109
Synthesis of optically active silyl protected cyanohydrins
1990 · J. Brussee, W.T. Loos, et al. · Tetrahedron · 108
2,4,6-Trisubstituted Pyrimidines as a New Class of Selective Adenosine A 1 Receptor Antagonists
2004 · Lisa C. W. Chang, Ronald F. Spanjersberg, et al. · Journal of Medicinal Chemistry · 102
The glutathione-binding site in glutathione S-transferases. Investigation of the cysteinyl, glycyl and γ-glutamyl domains
1990 · A E P Adang, J Brussee, et al. · Biochemical Journal · 99
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Effect of N-alkyl-azocycloheptan-2-ones including azone on the thermal behaviour of human stratum corneum
1989 · J.A. Bouwstra, L.J.C. Peschier, et al. · International Journal of Pharmaceutics · 96
Hybrid Ortho/Allosteric Ligands for the Adenosine A1Receptor
2010 · Rajeshwar Narlawar, J. Robert Lane, et al. · Journal of Medicinal Chemistry · 95
(β-Amino alcohol)(arene)ruthenium(II)-Catalyzed Asymmetric Transfer Hydrogenation of Functionalized Ketones − Scope, Isolation of the Catalytic Intermediates, and Deactivation Processes
2001 · Kathelyne Everaere, André Mortreux, et al. · European Journal of Organic Chemistry · 89
Visualisation of normal and enhanced HgCl2 transport through human skin in vitro
1989 · H.E. Boddé, M.A.M. Kruithof, et al. · International Journal of Pharmaceutics · 82
Kinetics, ultrastructural aspects and molecular modelling of transdermal peptide flux enhancement by N-alkylazacycloheptanones
1991 · A.J. Hoogstraate, J. Verhoef, et al. · International Journal of Pharmaceutics · 78
Synthesis of optically active ethanolamines.
1990 · J. Brussee, F. Dofferhoff, et al. · Tetrahedron · 73
Dual-Point Competition Association Assay: A Fast and High-Throughput Kinetic Screening Method for Assessing Ligand-Receptor Binding Kinetics
2012 · Dong Guo, Erika J.H. van Dorp, et al. · SLAS DISCOVERY · 67
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Hydroxynitrile lyases from almond and sorghum as biocatalysts
1991 · E. Smitskamp‐Wilms, J. Brussee, et al. · Recueil des Travaux Chimiques des Pays-Bas · 66
Magnesium ion mediated stereospecific formation of N-substituted ethanolamines during reductive amination
1990 · Johannes Brussee, Rolf A.T.M. van Benthem, et al. · Tetrahedron Asymmetry · 66
Structure–Kinetic Relationships—An Overlooked Parameter in Hit-to-Lead Optimization: A Case of Cyclopentylamines as Chemokine Receptor 2 Antagonists
2013 · Maris Vilums, Annelien J. M. Zweemer, et al. · Journal of Medicinal Chemistry · 65
False Positives in a Reporter Gene Assay: Identification and Synthesis of Substituted N-Pyridin-2-ylbenzamides as Competitive Inhibitors of Firefly Luciferase
2008 · Laura H. Heitman, Jacobus P. D. van Veldhoven, et al. · Journal of Medicinal Chemistry · 65
Works count: 151
Citation count: 5,086
H-index: 42
I10-index: 91
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