Product
Help
Pricing
About
Jobs
Log in
Get started
Author
Add to collection
Nikolaos Eleftheriadis
Observed names:
Eleftheriadis, Nikolaos,
Nicolaos Eleftheriadis
Institution:
University of Crete
Observed institutions:
University of Crete,
University of Groningen,
Aristotle University of Thessaloniki,
Rega Institute for Medical Research,
FORTH Institute of Molecular Biology and Biotechnology,
Zernike Institute for Advanced Materials,
Foundation for Research and Technology Hellas,
KU Leuven
show all 8
ORCID:
0000-0002-1738-6419
Observed ORCID:
0000-0002-1738-6419
OpenAlex ID:
A5078253777
Conformational and dynamic plasticity in substrate-binding proteins underlies selective transport in ABC importers
2019
·
Marijn de Boer
, Giorgos Gouridis
, et al.
·
eLife
·
133
HDAC1-3 inhibitor MS-275 enhances IL10 expression in RAW264.7 macrophages and reduces cigarette smoke-induced airway inflammation in mice
2017
·
Niek G. J. Leus
, Thea van den Bosch
, et al.
·
Scientific Reports
·
76
PDF
Rational Development of a Potent 15-Lipoxygenase-1 Inhibitor with in Vitro and ex Vivo Anti-inflammatory Properties
2015
·
Nikolaos Eleftheriadis
, Constantinos G. Neochoritis
, et al.
·
Journal of Medicinal Chemistry
·
56
Design of a novel thiophene inhibitor of 15-lipoxygenase-1 with both anti-inflammatory and neuroprotective properties
2016
·
Nikolaos Eleftheriadis
, Hessel Poelman
, et al.
·
European Journal of Medicinal Chemistry
·
50
PDF
On the impact of competing intra- and intermolecular triplet-state quenching on photobleaching and photoswitching kinetics of organic fluorophores
2018
·
Jochem H. Smit
, Jasper H. M. van der Velde
, et al.
·
Physical Chemistry Chemical Physics
·
46
PDF
Discovery of a novel activator of 5-lipoxygenase from an anacardic acid derived compound collection
2013
·
Rosalina Wisastra
, Petra A.M. Kok
, et al.
·
Bioorganic & Medicinal Chemistry
·
39
PDF
Identification of 6-benzyloxysalicylates as a novel class of inhibitors of 15-lipoxygenase-1
2015
·
Nikolaos Eleftheriadis
, Stephanie Thee
, et al.
·
European Journal of Medicinal Chemistry
·
34
PDF
One-pot microwave assisted synthesis of new 2-alkoxycarbonylmethylene-4-oxo-1,5-benzo-, naphtho-, and pyridodiazepines and assessment of their cytogenetic activity
2013
·
Nicolaos Eleftheriadis
, Constantinos G. Neochoritis
, et al.
·
European Journal of Medicinal Chemistry
·
34
Small Multitarget Molecules Incorporating the Enone Moiety
2019
·
Thalia Liargkova
, Nikolaos Eleftheriadis
, et al.
·
Molecules
·
26
PDF
A combinatorial approach for the discovery of drug-like inhibitors of 15-lipoxygenase-1
2019
·
Ramon van der Vlag
, Hao Guo
, et al.
·
European Journal of Medicinal Chemistry
·
25
PDF
Activity‐Based Probes for 15‐Lipoxygenase‐1
2016
·
Nikolaos Eleftheriadis
, Stephanie A. Thee
, et al.
·
Angewandte Chemie International Edition
·
24
Structural dynamics in the evolution of a bilobed protein scaffold
2021
·
Giorgos Gouridis
, Yusran A. Muthahari
, et al.
·
Proceedings of the National Academy of Sciences
·
22
PDF
Linker Molecules Convert Commercial Fluorophores into Tailored Functional Probes during Biolabelling
2022
·
Lei Zhang
, Michael Isselstein
, et al.
·
Angewandte Chemie International Edition
·
19
PDF
A nexus of intrinsic dynamics underlies translocase priming
2021
·
Srinath Krishnamurthy
, Nikolaos Eleftheriadis
, et al.
·
Structure
·
19
PDF
Discovery of chromenes as inhibitors of macrophage migration inhibitory factor
2017
·
Tjie Kok
, Hannah Wapenaar
, et al.
·
Bioorganic & Medicinal Chemistry
·
18
PDF
Ruthenium complexes as inhibitors of 15-lipoxygenase-1
2015
·
Katja Traven
, Nikolaos Eleftheriadis
, et al.
·
Polyhedron
·
18
PDF
Preproteins couple the intrinsic dynamics of SecA to its ATPase cycle to translocate via a catch and release mechanism
2022
·
Srinath Krishnamurthy
, Marios-Frantzeskos Sardis
, et al.
·
Cell Reports
·
15
PDF
A Trap-Door Mechanism for Zinc Acquisition by Streptococcus pneumoniae AdcA
2021
·
Zhenyao Luo
, Jacqueline R. Morey
, et al.
·
mBio
·
15
Identification of potential antivirulence agents by substitution-oriented screening for inhibitors of Streptococcus pyogenes sortase A
2018
·
Magdalena Wójcik
, Nikolaos Eleftheriadis
, et al.
·
European Journal of Medicinal Chemistry
·
13
PDF
Photoactivation provides a mechanistic explanation for pan-assay interference behaviour of 2-aminopyrroles in lipoxygenase inhibition
2017
·
Hao Guo
, Nikolaos Eleftheriadis
, et al.
·
European Journal of Medicinal Chemistry
·
13
A thorough study on the reaction of DMAD with 1-arylaminoimidazole-2-thiones. Expeditious synthesis of imidazo[2,1-b][1,3]thiazoles through a novel arylamino rearrangement
2009
·
Constantinos Neochoritis
, Nicolaos Eleftheriadis
, et al.
·
Tetrahedron
·
13
Investigating the Catalytic Site of Human 15‐Lipoxygenase‐1 via Marine Natural Products
2024
·
Ntaniela Spacho
, Marcello Casertano
, et al.
·
Chemistry - A European Journal
·
12
PDF
The relevance of K i calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor
2017
·
Hannah Wapenaar
, Thea van den Bosch
, et al.
·
European Journal of Medicinal Chemistry
·
11
PDF
One-Pot DBU-Promoted Synthesis of Hydroacridinones and Spirohexahydropyrimidines
2013
·
Julia Stephanidou-Stephanatou
, Constantinos Tsoleridis
, et al.
·
Synlett
·
7
The Evolution of Fluorescein into A Potential Theranostic Tool
2025
·
Konstantinos S. Adamis
, Michail Georgoulakis
, et al.
·
Chemistry - A European Journal
·
6
Show more works
View as search
Works count:
59
Citation count:
791
H-index:
16
I10-index:
23
Year
Topic
Type