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Syozo Kobayashi
Institution:
Daiichi-Sankyo (Japan)
Observed institution:
Daiichi-Sankyo (Japan)
OpenAlex ID:
A5084625618
Synthesis and Conformational Analysis of a Non-Amidine Factor Xa Inhibitor That Incorporates 5-Methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine as S4 Binding Element
2004
·
Noriyasu Haginoya
, Syozo Kobayashi
, et al.
·
Journal of Medicinal Chemistry
·
74
Discovery of N-[(1R,2S,5S)-2-{[(5-chloroindol-2-yl)carbonyl]amino}-5-(dimethylcarbamoyl)cyclohexyl]-5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxamide hydrochloride: A novel, potent and orally active direct inhibitor of factor Xa
2008
·
Tsutomu Nagata
, Toshiharu Yoshino
, et al.
·
Bioorganic & Medicinal Chemistry
·
43
Design, synthesis, and biological activity of non-amidine factor Xa inhibitors containing pyridine N-oxide and 2-carbamoylthiazole units
2004
·
Noriyasu Haginoya
, Syozo Kobayashi
, et al.
·
Bioorganic & Medicinal Chemistry
·
34
Orally active factor Xa inhibitors: 4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine derivatives
2004
·
Noriyasu Haginoya
, Syozo Kobayashi
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
19
Orally Active Factor Xa Inhibitors: 4,5,6,7‐Tetrahydrothiazolo[5,4‐c]pyridine Derivatives.
2004
·
Noriyasu Haginoya
, Syozo Kobayashi
, et al.
·
ChemInform
ChemInform Abstract: Novel Potassium Channel Opener Prodrugs with a Slow Onset and Prolonged Duration of Action.
2000
·
Haruhiko Horino
, Tetsuya Mimura
, et al.
·
ChemInform
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Works count:
6
Citation count:
170
H-index:
4
I10-index:
4
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