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Robert R. Wilkening

Observed names: R. R. WILKENING, R. R. Wilkening, R. Wilkening, R.R. Wilkening, ROBERT WILKENING, Robert Wilkening
OpenAlex ID: A5086657296
Conformational analysis of linear peptides: 5. Spectroscopic characterization of β-turns in Aib-containing oligopeptides in chloroform
1984 · Gian Maria Bonora, Claudio Mapelli, et al. · International Journal of Biological Macromolecules · 116
Ibrexafungerp: An orally active β-1,3-glucan synthesis inhibitor
2020 · James M. Apgar, Robert R. Wilkening, et al. · Bioorganic & Medicinal Chemistry Letters · 55
An efficient synthesis of 2-substituted-thio-6-hydroxyethyl-penem-3-carboxylic acids via 2-thioxopenams
1983 · W.J. Leanza, Frank DiNinno, et al. · Tetrahedron · 49
The discovery of tetrahydrofluorenones as a new class of estrogen receptor β-subtype selective ligands
2006 · R.R. Wilkening, R.W. Ratcliffe, et al. · Bioorganic & Medicinal Chemistry Letters · 44
Pharmacological AMPK activation induces transcriptional responses congruent to exercise in skeletal and cardiac muscle, adipose tissues and liver
2019 · Eric S. Muise, Hong-Ping Guan, et al. · PLoS ONE · 41
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Selective estrogen receptor-beta (SERM-beta) compounds modulate raphe nuclei tryptophan hydroxylase-1 (TPH-1) mRNA expression and cause antidepressant-like effects in the forced swim test
2012 · J.A. Clark, S. Alves, et al. · Neuropharmacology · 40
Reduced Immunotoxicity and Preservation of Antibacterial Activity in a Releasable Side-Chain Carbapenem Antibiotic
1999 · Hugh Rosen, Richard Hajdu, et al. · Science · 37
Synthesis and biological evaluation of antifungal derivatives of enfumafungin as orally bioavailable inhibitors of β-1,3-glucan synthase
2012 · Brian H. Heasley, Gregory J. Pacofsky, et al. · Bioorganic & Medicinal Chemistry Letters · 35
The synthesis of novel 8a-aza-8a-homoerythromycin derivatives via the beckmann rearrangement of (9z)-erythromycin a oxime
1993 · Robert R. Wilkening, Ronald W. Ratcliffe, et al. · Bioorganic & Medicinal Chemistry Letters · 35
Novel orally active inhibitors of β-1,3-glucan synthesis derived from enfumafungin
2015 · James M. Apgar, Robert R. Wilkening, et al. · Bioorganic & Medicinal Chemistry Letters · 34
Estrogen receptor β-subtype selective tetrahydrofluorenones: Use of a fused pyrazole as a phenol bioisostere
2006 · R.R. Wilkening, R.W. Ratcliffe, et al. · Bioorganic & Medicinal Chemistry Letters · 34
Synthesis and activity of 2-(sulfonamido)methyl-carbapenems: Discovery of a novel, anti-MRSA 1,8-naphthosultam pharmacophore
1999 · R.R. Wilkening, R.W. Ratcliffe, et al. · Bioorganic & Medicinal Chemistry Letters · 32
Synthesis and properties of 2-(naphthosultamyl)methyl-carbapenems with potent anti-MRSA activity: Discovery of L-786,392
1999 · R.W. Ratcliffe, R.R. Wilkening, et al. · Bioorganic & Medicinal Chemistry Letters · 29
Conformational analysis of linear peptides. 4. Association properties of protected oligomers of .alpha.-aminoisobutyric acid in chloroform
1983 · Robert R. Wilkening, E. S. Stevens, et al. · Journal of the American Chemical Society · 22
Structure–activity-relationship of amide and sulfonamide analogs of omarigliptin
2015 · Ping Chen, Dennis Feng, et al. · Bioorganic & Medicinal Chemistry Letters · 20
Triazolo-tetrahydrofluorenones as selective estrogen receptor beta agonists
2006 · Dann L. Parker, Dongfang Meng, et al. · Bioorganic & Medicinal Chemistry Letters · 20
Benzothiazolylthio carbapenems: potent anti-MRSA agents
1995 · Sherman T. Waddell, Ronald W. Ratcliffe, et al. · Bioorganic & Medicinal Chemistry Letters · 19
Control of rat tail skin temperature regulation by estrogen receptor-beta selective ligand
2009 · Evan E. Opas, Angela Scafonas, et al. · Maturitas · 17
In vivo Evaluation of Three Acid-stable Azalide Compounds, L-701,677, L-708,299 and L-708,365 Compared to Erythromycin, Azithromycin and Clarithromycin.
1995 · CHARLES J. GILL, GEORGE K. ABRUZZO, et al. · The Journal of Antibiotics · 9
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ChemInform Abstract: CONFORMATIONAL ANALYSIS OF LINEAR PEPTIDES. 4. ASSOCIATION PROPERTIES OF PROTECTED OLIGOMERS OF α‐AMINOISOBUTYRIC ACID IN CHLOROFORM
1983 · R. R. WILKENING, E. S. STEVENS, et al. · ChemInform · 9
Novel transannular rearrangements of azalide iminoethers
1997 · Robert R. Wilkening, Ronald W. Ratcliffe, et al. · Tetrahedron · 8
MK-5204: An orally active β-1,3-glucan synthesis inhibitor
2020 · James M. Apgar, Robert R. Wilkening, et al. · Bioorganic & Medicinal Chemistry Letters · 7
Preparation and activities of 4″-epi and 4″-deoxy-4″-amino analogs derived from 9-deoxo-8a-aza-8a-homoerythromycin A
1994 · K. Shankaran, Robert R. Wilkening, et al. · Bioorganic & Medicinal Chemistry Letters · 7
Erratum to “Triazolo-tetrahydrofluorenones as selective estrogen receptor beta agonists” [Bioorg. Med. Chem. Lett. 16 (2006) 4652–4656]
2006 · Dann L. Parker, Dongfang Meng, et al. · Bioorganic & Medicinal Chemistry Letters · 1
Estrogen Receptor β‐Subtype Selective Tetrahydrofluorenones: Use of a Fused Pyrazole as a Phenol Bioisostere.
2006 · R. R. Wilkening, et al. et al. · ChemInform
Works count: 29
Citation count: 720
H-index: 17
I10-index: 18
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