Get started
Author

Nicolas Boutard

Peptide Scanning for Studying Structure‐Activity Relationships in Drug Discovery
2012 · Andrew G. Jamieson, Nicolas Boutard, et al. · Chemical Biology & Drug Design · 98
Positional Scanning for Peptide Secondary Structure by Systematic Solid-Phase Synthesis of Amino Lactam Peptides
2009 · Andrew G. Jamieson, Nicolas Boutard, et al. · Journal of the American Chemical Society · 82
Synthetic Lethality Triggered by Combining Olaparib with BRCA2–Rad51 Disruptors
2017 · Federico Falchi, Elisa Giacomini, et al. · ACS Chemical Biology · 47
PDF
β,β-Disubstituted C- and N-Vinylindoles from One-Step Condensations of Aldehydes and Indole Derivatives
2009 · Gil Fridkin, Nicolas Boutard, et al. · The Journal of Organic Chemistry · 47
Discovery of a series of ester-substituted NLRP3 inflammasome inhibitors
2020 · David Harrison, Nicolas Boutard, et al. · Bioorganic & Medicinal Chemistry Letters · 40
Structure–Activity Analysis of the Growth Hormone Secretagogue GHRP‐6 by α‐ and β‐Amino γ‐Lactam Positional Scanning
2009 · Nicolas Boutard, Andrew G. Jamieson, et al. · Chemical Biology & Drug Design · 33
Synthesis of amide and sulfonamide substituted N-aryl 6-aminoquinoxalines as PFKFB3 inhibitors with improved physicochemical properties
2018 · Nicolas Boutard, Arkadiusz Białas, et al. · Bioorganic & Medicinal Chemistry Letters · 23
Discovery and Structure–Activity Relationships of N‐Aryl 6‐Aminoquinoxalines as Potent PFKFB3 Kinase Inhibitors
2018 · Nicolas Boutard, Arkadiusz Białas, et al. · ChemMedChem · 21
Examination of the active secondary structure of the peptide 101.10, an allosteric modulator of the interleukin‐1 receptor, by positional scanning using β‐amino γ‐lactams
2011 · Nicolas Boutard, Stéphane Turcotte, et al. · Journal of Peptide Science · 18
Pyrrolo[3,2-e][1,4]diazepin-2-one Synthesis: A Head-to-Head Comparison of Soluble versus Insoluble Supports
2011 · Nicolas Boutard, Julien Dufour-Gallant, et al. · The Journal of Organic Chemistry · 15
Easy saponification by metal silanolates: application in SPPS and in (S)-5-hydroxynorvaline preparation
2005 · Ewelina Minta, Cédric Boutonnet, et al. · Tetrahedron Letters · 15
5-Keto-3-cyano-2,4-diaminothiophenes as selective maternal embryonic leucine zipper kinase inhibitors
2018 · Nicolas Boutard, Aleksandra Sabiniarz, et al. · Bioorganic & Medicinal Chemistry Letters · 9
NewC-Glycosylated α -Amino Acid Synthesis by Addition Reaction of an Amino Acid Organozinc Reagent on Carbohydrate-Derived Aldehydes
2012 · Nicolas Boutard, Frédéric Labéguère, et al. · Synthetic Communications · 4
Abstract 1806: Discovery of novel MTA-cooperative PRMT5 inhibitors as a targeted therapeutics for MTAP deleted cancers
2022 · Oleksandr Levenets, Anna Bartosik, et al. · Cancer Research · 2
Abstract 3516: Discovery of novel SHMT small molecule inhibitors for cancer treatment
2018 · Anna Bartosik, Pawel Guzik, et al. · Cancer Research · 2
Abstract 4598: Discovery of novel MTA-cooperative PRMT5 inhibitors as targeted therapeutics for MTAP-deleted cancers
2024 · Adam Radzimierski, Aneta Bobowska, et al. · Cancer Research · 1
Abstract 1281: Development and characterization of small molecule HPK1 inhibitors
2021 · Maciej Kujawa, Eliza Zimoląg, et al. · Cancer Research · 1
9.13.5 1H-Pyrroles (Update 2013)
2013 · W. D. Lubell, D. J. St-Cyr, et al. · Haug Verlag in Georg Thieme Verlag KG eBooks · 1
Abstract C135: Discovery of novel MTA-cooperative PRMT5 inhibitors as targeted therapeutics for MTAP-deleted cancers
2023 · Adam Radzimierski, Aneta Bobowska, et al. · Molecular Cancer Therapeutics
Abstract 449: Discovery of novel MTA-cooperative PRMT5 inhibitors as targeted therapeutics for MTAP-deleted cancers
2023 · Anna Bartosik, Adam Radzimierski, et al. · Cancer Research
Discovery of novel MTA-cooperative PRMT5 inhibitors as targeted therapeutics for MTAP deleted cancers
2022 · A. Bartosik, A. Radzimierski, et al. · European Journal of Cancer
PDF
Knowledge Updates 2013/1
2013 · A. Fuerstner, K. Ishihara, et al. · Haug Verlag in Georg Thieme Verlag KG eBooks
ChemInform Abstract: New C‐Glycosylated α‐Amino Acid Synthesis by Addition Reaction of an Amino Acid Organozinc Reagent on Carbohydrate‐Derived Aldehydes.
2012 · Nicolas Boutard, Frederic Labeguere, et al. · ChemInform
CCDC 717034: Experimental Crystal Structure Determination
2010 · Fridkin, G., Boutard, N., et al. · The Cambridge Structural Database
ChemInform Abstract: β,β‐Disubstituted C‐ and N‐Vinylindoles from One‐Step Condensations of Aldehydes and Indole Derivatives.
2009 · Gil Fridkin, Nicolas Boutard, et al. · ChemInform
Works count: 27
Citation count: 459
H-index: 11
I10-index: 11
Year
Topic
Type