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Nagaaki Sato

Observed names: N Sato, N. SATO, N. Sato, Naga‐aki Sato, Sato, Nagaaki
OpenAlex ID: A5111593751
Development of a selective and potent radioactive ligand for histamine H3 receptors: A compound potentially useful for receptor occupancy studies
2009 · Yuko Mitobe, Sayaka Ito, et al. · Bioorganic & Medicinal Chemistry Letters · 80
A neuropeptide Y Y5 antagonist selectively ameliorates body weight gain and associated parameters in diet-induced obese mice
2006 · Akane Ishihara, Akio Kanatani, et al. · Proceedings of the National Academy of Sciences · 76
Total Synthesis of Octalactin A and B
1994 · Keith R. Buszek, Nagaaki Sato, et al. · Journal of the American Chemical Society · 72
Synthesis, Structure−Activity Relationships, and Biological Profiles of a Quinazolinone Class of Histamine H3Receptor Inverse Agonists
2008 · Tsuyoshi Nagase, Takashi Mizutani, et al. · Journal of Medicinal Chemistry · 71
Facile One-Pot Synthesis of N -Difluoromethyl-2-pyridone Derivatives
2006 · Makoto Ando, Toshihiro Wada, et al. · Organic Letters · 70
Modulation of neuropeptide Y receptors for the treatment of obesity
2009 · Nagaaki Sato, Yoshio Ogino, et al. · Expert Opinion on Therapeutic Patents · 60
(9S)-9-(2-Hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one, a Selective and Orally Active Neuropeptide Y Y5 Receptor Antagonist
2008 · Nagaaki Sato, Makoto Jitsuoka, et al. · Journal of Medicinal Chemistry · 59
Inverse agonist histamine H3 receptor PET tracers labelled with carbon‐11 or fluorine‐18
2009 · Terence G. Hamill, Nagaaki Sato, et al. · Synapse · 45
Synthesis and Evaluation of a Novel Indoledione Class of Long Chain Fatty Acid Elongase 6 (ELOVL6) Inhibitors
2009 · Toshiyuki Takahashi, Tsuyoshi Nagase, et al. · Journal of Medicinal Chemistry · 43
Total synthesis of octalactin A via ring-closing metathesis reaction
2002 · Keith R Buszek, Nagaaki Sato, et al. · Tetrahedron Letters · 43
Mechanism of the anti‐obesity effects induced by a novel Melanin‐concentrating hormone 1‐receptor antagonist in mice
2009 · Masahiko Ito, A Ishihara, et al. · British Journal of Pharmacology · 38
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Design and Synthesis of the Potent, Orally Available, Brain-Penetrable Arylpyrazole Class of Neuropeptide Y5 Receptor Antagonists
2003 · Nagaaki Sato, Toshiyuki Takahashi, et al. · Journal of Medicinal Chemistry · 38
Synthesis, characterization, and monkey positron emission tomography (PET) studies of [18F]Y1-973, a PET tracer for the neuropeptide Y Y1 receptor
2010 · Eric D. Hostetler, Sandra Sanabria-Bohórquez, et al. · NeuroImage · 35
Novel potent neuropeptide Y Y5 receptor antagonists: Synthesis and structure–activity relationships of phenylpiperazine derivatives
2006 · Toshiyuki Takahashi, Aya Sakuraba, et al. · Bioorganic & Medicinal Chemistry · 33
Development of novel 2-[4-(aminoalkoxy)phenyl]-4(3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists
2008 · Takashi Mizutani, Tsuyoshi Nagase, et al. · Bioorganic & Medicinal Chemistry Letters · 32
Blockade of body weight gain and plasma corticosterone levels in Zucker fatty rats using an orally active neuropeptide Y Y1 antagonist
2002 · Akane Ishihara, Akio Kanatani, et al. · British Journal of Pharmacology · 29
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Discovery of Tetrasubstituted Imidazolines as Potent and Selective Neuropeptide Y Y5 Receptor Antagonists: Reduced Human Ether-a-go-go Related Gene Potassium Channel Binding Affinity and Potent Antiobesity Effect
2009 · Nagaaki Sato, Makoto Ando, et al. · Journal of Medicinal Chemistry · 28
Discovery of pyridone-containing imidazolines as potent and selective inhibitors of neuropeptide Y Y5 receptor
2009 · Makoto Ando, Nagaaki Sato, et al. · Bioorganic & Medicinal Chemistry · 26
Facile Synthesis of Saturated Eight-membered Ring Lactones
2001 · Keith R. Buszek, Youngmee Jeong, et al. · Synthetic Communications · 25
Discovery and characterization of a novel potent, selective and orally active inhibitor for mammalian ELOVL6
2010 · Ken Shimamura, Akira Nagumo, et al. · European Journal of Pharmacology · 23
Discovery of Novel Benzoxazinones as Potent and Orally Active Long Chain Fatty Acid Elongase 6 Inhibitors
2009 · Takashi Mizutani, Shiho Ishikawa, et al. · Journal of Medicinal Chemistry · 22
The effects of a novel histamine-3 receptor inverse agonist on essential tremor in comparison to stable levels of alcohol
2011 · RWM Zoethout, R Iannone, et al. · Journal of Psychopharmacology · 20
Melanin-concentrating hormone 1-receptor antagonist suppresses body weight gain correlated with high receptor occupancy levels in diet-induced obesity mice
2009 · Masahiko Ito, Akane Ishihara, et al. · European Journal of Pharmacology · 20
Discovery of novel spiro-piperidine derivatives as highly potent and selective melanin-concentrating hormone 1 receptor antagonists
2009 · Takao Suzuki, Minoru Moriya, et al. · Bioorganic & Medicinal Chemistry Letters · 20
Discovery of substituted 2,4,4-triarylimidazoline derivatives as potent and selective neuropeptide Y Y5 receptor antagonists
2009 · Nagaaki Sato, Makoto Jitsuoka, et al. · Bioorganic & Medicinal Chemistry Letters · 20
Works count: 58
Citation count: 1,235
H-index: 21
I10-index: 36
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