Author

Jan W. F. Wasley

Observed names: J W Wasley, J WASLEY, J. W. F. WASLEY, J. W. F. Wasley, J. Wasley, J.W.F. Wasley, Jan W.F Wasley, Jan W.F. Wasley, Jan Wasley

Observed institution: National Research Council Canada

OpenAlex ID: A5111823698

Biochemical and pharmacological characterization of CGS 12066B, a selective serotonin-1B agonist

1987 · Robert F. Neale, Scott L. Fallon, et al. · European Journal of Pharmacology · 160

.beta.-Lapachone: synthesis of derivatives and activities in tumor models

1984 · Karl Schaffner-Sabba, Karl H. Schmidt-Ruppin, et al. · Journal of Medicinal Chemistry · 116

CGS 9343B, a novel, potent, and selective inhibitor of calmodulin activity.

1987 · J A Norman, J Ansell, et al. · Molecular Pharmacology · 107

Imidazo[1,5-a]pyridines: a new class of thromboxane A2 synthetase inhibitors

1985 · Neville F. Ford, Leslie J. Browne, et al. · Journal of Medicinal Chemistry · 106

NGB 2904 and NGB 2849: Two highly selective dopamine D3 receptor antagonists

1998 · Jun Yuan, Xi Chen, et al. · Bioorganic & Medicinal Chemistry Letters · 75

Discovery of S-Nitrosoglutathione Reductase Inhibitors: Potential Agents for the Treatment of Asthma and Other Inflammatory Diseases

2011 · Xicheng Sun, Jan W. F. Wasley, et al. · ACS Medicinal Chemistry Letters · 59

2-Phenyl-4(5)-[[4-(pyrimidin-2- yl)piperazin-1-yl]methyl]imidazole. A Highly Selective Antagonist at Cloned Human D 4 Receptors

1997 · Andrew Thurkauf, Jun Yuan, et al. · Journal of Medicinal Chemistry · 58

Indoline and piperazine containing derivatives as a novel class of mixed D2/D4 receptor antagonists. Part 2: Asymmetric synthesis and biological evaluation

2002 · He Zhao, Xiaoshu He, et al. · Bioorganic & Medicinal Chemistry Letters · 56

Structures of Chlorobium Chlorophylls (660)

1966 · A. S. Holt, J. W. Purdie, et al. · Canadian Journal of Chemistry · 52

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trans-1-[(2-Phenylcyclopropyl)methyl]-4-arylpiperazines: Mixed Dopamine D2/D4 Receptor Antagonists as Potential Antipsychotic Agents

2000 · Xiaoyan Zhang, Kevin Hodgetts, et al. · Journal of Medicinal Chemistry · 36

1-Phenyl-3-(aminomethyl)pyrroles as Potential Antipsychotic Agents. Synthesis and Dopamine Receptor Binding

1995 · Andrew Thurkauf, Jun Yuan, et al. · Journal of Medicinal Chemistry · 36

56. 2,2′-Bipyrroles

1963 · R. Grigg, A. W. Johnson, et al. · Journal of the Chemical Society (Resumed) · 31

Discovery of potent and novel S-nitrosoglutathione reductase inhibitors devoid of cytochrome P450 activities

2011 · Xicheng Sun, Jian Qiu, et al. · Bioorganic & Medicinal Chemistry Letters · 29

Characterization of CGS 8515 as a selective 5-lipoxygenase inhibitor using in vitro and in vivo models

1988 · Edmond C. Ku, Anil Raychaudhuri, et al. · Biochimica et Biophysica Acta (BBA) - Lipids and Lipid Metabolism · 25

Structure–activity relationships of pyrrole based S-nitrosoglutathione reductase inhibitors: Pyrrole regioisomers and propionic acid replacement

2011 · Xicheng Sun, Jian Qiu, et al. · Bioorganic & Medicinal Chemistry Letters · 24

Indoline and piperazine containing derivatives as a novel class of mixed D2/D4 receptor antagonists. Part 1: Identification and structure–activity relationships

2002 · He Zhao, Andrew Thurkauf, et al. · Bioorganic & Medicinal Chemistry Letters · 24

Novel calmodulin antagonist CGS 9343B inhibits secretory diarrhea.

1989 · J E Shook, T F Burks, et al. · Journal of Pharmacology and Experimental Therapeutics · 23

A practical synthesis of 1,3,4,14b‐tetrahydro‐2‐methyl‐10H‐pyrazino‐[1,2‐a]pyrrolo[2,1‐c][1,4]benzodiazepine (1:1) maleate

1984 · S. K. Boyer, G. Fitchett, et al. · Journal of Heterocyclic Chemistry · 21

Synthesis of 1-Arylsulfonylpyrroles

1973 · Jan W. F. Wasley, Kenneth Chan · Synthetic Communications · 20

CMorophyllides c

1970 · J. W. F. Wasley, W. T. Scott, et al. · Canadian Journal of Biochemistry · 20

431. The condensation of 2,2′-bipyrroles with 2-formylpyrroles and 5,5′-diformyldipyrromethanes

1963 · E. Bullock, R. Grigg, et al. · Journal of the Chemical Society (Resumed) · 20

Medicinal chemistry education: what is needed and where is it going?

2005 · Povl Krogsgaard‐Larsen, Roberto Pelliciari, et al. · Drug Development Research · 19

CGS 20625, a novel pyrazolopyridine anxiolytic.

1989 · M Williams, D A Bennett, et al. · Journal of Pharmacology and Experimental Therapeutics · 19

6-(4-Benzylpiperazin-1-yl)benzodioxanes as selective ligands at cloned primate dopamine D4 receptors

2001 · Kevin J Hodgetts, Andrzej Kieltyka, et al. · Bioorganic & Medicinal Chemistry · 18

Synthesis of 1-Substituted Pyrrole-3-carboxaldehydes

1983 · Ali Hamdan, Jan W. F. Wasley · Synthetic Communications · 18

Works count: 69

Citation count: 1,313

H-index: 20

I10-index: 33