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Richard Saperstein

Observed names: R Saperstein, R. SAPERSTEIN, R. Saperstein, RICHARD SAPERSTEIN
OpenAlex ID: A5111833873
A potent cyclic hexapeptide analogue of somatostatin
1981 · Daniel F. Veber, Roger M. Freidinger, et al. · Nature · 419
Thiazolidinediones produce a conformational change in peroxisomal proliferator-activated receptor-gamma: binding and activation correlate with antidiabetic actions in db/db mice
1996 · J Berger, P Bailey, et al. · Endocrinology · 391
Bioactive Conformation of Luteinizing Hormone-Releasing Hormone: Evidence from a Conformationally Constrained Analog
1980 · Roger M. Freidinger, Daniel F. Veber, et al. · Science · 315
Decreased expression of the insulin-responsive glucose transporter in diabetes and fasting
1989 · Joel Berger, Chhabi Biswas, et al. · Nature · 299
Highly active cyclic and bicyclic somatostatin analogues of reduced ring size
1979 · DANIEL F. VEBER, FREDERICK W. HOLLY, et al. · Nature · 213
The Isolation and Metabolism of Brown Fat Cells
1967 · John N. Fain, Nora Reed, et al. · Journal of Biological Chemistry · 171
A super active cyclic hexapeptide analog of somatostatin
1984 · Daniel F. Veber, Richard Saperstein, et al. · Life Sciences · 165
Conformationally restricted bicyclic analogs of somatostatin.
1978 · D F Veber, F W Holly, et al. · Proceedings of the National Academy of Sciences · 144
Hypothalamic Hormones
1976 · S Reichlin, R Saperstein, et al. · Annual Review of Physiology · 142
A selective human beta3 adrenergic receptor agonist increases metabolic rate in rhesus monkeys.
1998 · M H Fisher, A M Amend, et al. · Journal of Clinical Investigation · 116
A Novel Glucagon Receptor Antagonist Inhibits Glucagon-Mediated Biological Effects
2004 · Sajjad A. Qureshi, Mari Rios Candelore, et al. · Diabetes · 109
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Design of a selective insulin receptor tyrosine kinase inhibitor and its effect on glucose uptake and metabolism in intact cells
1989 · Richard Saperstein, Pasquale P. Vicario, et al. · Biochemistry · 108
The Insulin-Mimetic Effect of Vanadate Is Not Correlated with Insulin Receptor Tyrosine Kinase Activity Nor Phosphorylation in Mouse Diaphragmin Vivo
1989 · H. V. STROUT, P. P. VICARIO, et al. · Endocrinology · 108
Vanadate Treatment of Streptozotocin Diabetic Rats Restores Expression of the Insulin-Responsive Glucose Transporter in Skeletal Muscle
1990 · H. VINCENT STROUT, PASQUALE P. VICARIO, et al. · Endocrinology · 76
Nonreducible cyclic analogues of somatostatin
1976 · Daniel F. Veber, Robert G. Strachan, et al. · Journal of the American Chemical Society · 72
Serum Half-Life and Biological Activity of Mutants of Human Insulin-Like Growth Factor I which Do Not Bind to Serum Binding Proteins
1988 · MARGARET A. CASCIERI, RICHARD SAPERSTEIN, et al. · Endocrinology · 69
Activation of Insulin Signal Transduction Pathway and Anti-diabetic Activity of Small Molecule Insulin Receptor Activators
2000 · Sajjad A. Qureshi, Victor Ding, et al. · Journal of Biological Chemistry · 67
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Synthesis of nonreducible bicyclic analogs of somatostatin
1980 · Ruth F. Nutt, Daniel F. Veber, et al. · Journal of the American Chemical Society · 61
Conformational modifications of cyclic hexapeptide somatostatin analogs
1984 · Roger M. Freidinger, Debra Schwenk Perlow, et al. · International journal of peptide & protein research · 59
Discovery and investigation of a novel class of thiophene-derived antagonists of the human glucagon receptor
2005 · Joseph L. Duffy, Brian A. Kirk, et al. · Bioorganic & Medicinal Chemistry Letters · 57
Approaches to peptidomimetics which serve as surrogates for the cis amide bond: novel disulfide-constrained bicyclic hexapeptide analogs of somatostatic.
1993 · Stephen F. Brady, William J. Paleveda, et al. · Tetrahedron · 52
Discovery of novel, potent, selective, and orally active human glucagon receptor antagonists containing a pyrazole core
2010 · Dong-Ming Shen, Edward J. Brady, et al. · Bioorganic & Medicinal Chemistry Letters · 47
Synthesis and hypoglycemic activity of substituted 8-(1-piperazinyl)imidazo[1,2-a]pyrazines
1992 · Laura C. Meurer, Richard L. Tolman, et al. · Journal of Medicinal Chemistry · 45
Discovery of novel, potent, and orally active spiro-urea human glucagon receptor antagonists
2005 · Dong-Ming Shen, Fengqi Zhang, et al. · Bioorganic & Medicinal Chemistry Letters · 40
Hepatic glucagon receptor binding and glucose-lowering in vivo by peptidyl and non-peptidyl glucagon receptor antagonists
2004 · Qing Dallas-Yang, Xiaolan Shen, et al. · European Journal of Pharmacology · 40
Works count: 64
Citation count: 3,884
H-index: 30
I10-index: 43
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