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Rei Okamoto

Small molecule inhibition of cGAS reduces interferon expression in primary macrophages from autoimmune mice
2017 · Jessica Vincent, Carolina Adura, et al. · Nature Communications · 395
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Development of human cGAS-specific small-molecule inhibitors for repression of dsDNA-triggered interferon expression
2019 · Lodoe Lama, Carolina Adura, et al. · Nature Communications · 315
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Antimalarial proteasome inhibitor reveals collateral sensitivity from intersubunit interactions and fitness cost of resistance
2018 · Laura A. Kirkman, Wenhu Zhan, et al. · Proceedings of the National Academy of Sciences · 103
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Simple Construction of Bicyclo[4.3.0]nonane, Bicyclo[3.3.0]octane, and Related Benzo Derivatives by Palladium-Catalyzed Cycloalkenylation
2002 · Masahiro Toyota, Andivelu Ilangovan, et al. · Organic Letters · 65
Development of a Highly Selective Plasmodium falciparum Proteasome Inhibitor with Anti‐malaria Activity in Humanized Mice
2021 · Wenhu Zhan, Hao Zhang, et al. · Angewandte Chemie International Edition · 46
Novel Pure αVβ3 Integrin Antagonists That Do Not Induce Receptor Extension, Prime the Receptor, or Enhance Angiogenesis at Low Concentrations
2019 · Jihong Li, Yoshiyuki Fukase, et al. · ACS Pharmacology & Translational Science · 40
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Toward the Total Synthesis of (±)-Andrastin C
2012 · Rei Okamoto, Kazutaka Takeda, et al. · The Journal of Organic Chemistry · 31
Publisher Correction: Small molecule inhibition of cGAS reduces interferon expression in primary macrophages from autoimmune mice
2017 · Jessica Vincent, Carolina Adura, et al. · Nature Communications · 26
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Discovery and characterization of selective human sphingomyelin synthase 2 inhibitors
2017 · Ryutaro Adachi, Kazumasa Ogawa, et al. · European Journal of Medicinal Chemistry · 26
Design, Synthesis, and Optimization of Macrocyclic Peptides as Species-Selective Antimalaria Proteasome Inhibitors
2022 · Hao Zhang, John Ginn, et al. · Journal of Medicinal Chemistry · 25
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Selective Phenylimidazole-Based Inhibitors of the Mycobacterium tuberculosis Proteasome
2019 · Wenhu Zhan, Hao-Chi Hsu, et al. · Journal of Medicinal Chemistry · 22
Macrocyclic Peptides that Selectively Inhibit the Mycobacterium tuberculosis Proteasome
2021 · Hao Zhang, Hao-Chi Hsu, et al. · Journal of Medicinal Chemistry · 19
Structure–Activity Relationship Studies of Antimalarial Plasmodium Proteasome Inhibitors─Part II
2023 · Hao Zhang, John Ginn, et al. · Journal of Medicinal Chemistry · 18
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Discovery of 3,5-Diphenyl-4-methyl-1,3-oxazolidin-2-ones as Novel, Potent, and Orally Available Δ-5 Desaturase (D5D) Inhibitors
2017 · Jun Fujimoto, Rei Okamoto, et al. · Journal of Medicinal Chemistry · 18
Discovery of 1,8-naphthyridin-2-one derivative as a potent and selective sphingomyelin synthase 2 inhibitor
2020 · Takafumi Yukawa, Takashi Nakahata, et al. · Bioorganic & Medicinal Chemistry · 11
Structure‐Based Design, Synthesis, and Biological Evaluation of Imidazo[4,5‐b]pyridin‐2‐one‐Based p38 MAP Kinase Inhibitors: Part 1
2019 · Akira Kaieda, Masashi Takahashi, et al. · ChemMedChem · 10
Whole Cell Active Inhibitors of Mycobacterial Lipoamide Dehydrogenase Afford Selectivity over the Human Enzyme through Tight Binding Interactions
2021 · John Ginn, Xiuju Jiang, et al. · ACS Infectious Diseases · 8
Development of a Highly Selective Plasmodium falciparum Proteasome Inhibitor with Anti‐malaria Activity in Humanized Mice
2021 · Wenhu Zhan, Hao Zhang, et al. · Angewandte Chemie · 6
Structure‐Based Design, Synthesis, and Biological Evaluation of Imidazo[4,5‐b]Pyridin‐2‐one‐Based p38 MAP Kinase Inhibitors: Part 2
2019 · Akira Kaieda, Masashi Takahashi, et al. · ChemMedChem · 6
Ti(III)-induced radical cyclization. A stereoselective entry to the perhydrobenzo[e]indene unit of new protein farnesyltransferase inhibitors, andrastins A–D
2004 · Masahiro Toyota, Rei Okamoto, et al. · Tetrahedron Letters · 6
Structure–Activity Relationship Study of Antimalarial Asparagine-Derived Proteasome Inhibitors
2026 · Hao Zhang, Daqiang Li, et al. · ACS Omega
CCDC 1968615: Experimental Crystal Structure Determination
2020 · Yukawa, Takafumi, Nakahata, Takashi, et al. · The Cambridge Structural Database
CCDC 1519191: Experimental Crystal Structure Determination
2017 · Fujimoto, Jun, Okamoto, Rei, et al. · The Cambridge Structural Database
Ti(III)‐Induced Radical Cyclization. A Stereoselective Entry to the Perhydrobenzo[e]indene Unit of New Protein Farnesyltransferase Inhibitors, Andrastins A—D.
2005 · Masahiro Toyota, Rei Okamoto, et al. · ChemInform
Simple Construction of Bicyclo[4.3.0]nonane, Bicyclo[3.3.0]octane, and Related Benzo Derivatives by Palladium‐Catalyzed Cycloalkenylation.
2003 · Masahiro Toyota, Andivelu Ilangovan, et al. · ChemInform
Works count: 25
Citation count: 1,196
H-index: 14
I10-index: 16
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