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Masahiro Fuji
Observed names:
Fuji, Masahiro,
M Fuji,
M. FUJI,
MASAHIRO FUJI,
Masahiro FUJI,
冨士雅弘,
雅弘 冨士
show all 7
Institution:
Shionogi (Japan)
Observed institutions:
Shionogi (Japan),
Stanford University,
The University of Osaka
OpenAlex ID:
A5113213826
Highly Selective and Orally Active Inhibitors of Type IV Collagenase (MMP-9 and MMP-2): N-Sulfonylamino Acid Derivatives
1998
·
Yoshinori Tamura
, Fumihiko Watanabe
, et al.
·
Journal of Medicinal Chemistry
·
286
Carbamoyl Pyridone HIV-1 Integrase Inhibitors 3. A Diastereomeric Approach to Chiral Nonracemic Tricyclic Ring Systems and the Discovery of Dolutegravir (S/GSK1349572) and (S/GSK1265744)
2013
·
Brian A. Johns
, Takashi Kawasuji
, et al.
·
Journal of Medicinal Chemistry
·
190
The Transition Metal-Catalyzed Intermolecular [5+2] Cycloaddition: The Homologous Diels−Alder Reaction
1998
·
Paul A. Wender
, Heiko Rieck
, et al.
·
Journal of the American Chemical Society
·
155
Rhodium-Catalyzed [5 + 2] Cycloadditions of Allenes and Vinylcyclopropanes: Asymmetric Total Synthesis of (+)-Dictamnol
1999
·
Paul A. Wender
, Masahiro Fuji
, et al.
·
Organic Letters
·
127
Carbamoyl Pyridone HIV-1 Integrase Inhibitors. 2. Bi- and Tricyclic Derivatives Result in Superior Antiviral and Pharmacokinetic Profiles
2013
·
Takashi Kawasuji
, Brian A. Johns
, et al.
·
Journal of Medicinal Chemistry
·
97
A platform for designing HIV integrase inhibitors. Part 2: A two-metal binding model as a potential mechanism of HIV integrase inhibitors
2006
·
Takashi Kawasuji
, Masahiro Fuji
, et al.
·
Bioorganic & Medicinal Chemistry
·
88
3-Hydroxy-1,5-dihydro-pyrrol-2-one derivatives as advanced inhibitors of HIV integrase
2007
·
Takashi Kawasuji
, Masahiro Fuji
, et al.
·
Bioorganic & Medicinal Chemistry
·
75
Carbamoyl Pyridone HIV-1 Integrase Inhibitors. 1. Molecular Design and Establishment of an Advanced Two-Metal Binding Pharmacophore
2012
·
Takashi Kawasuji
, Brian A. Johns
, et al.
·
Journal of Medicinal Chemistry
·
61
Total Synthesis of Terprenin, a Novel Immunosuppressive p-Terphenyl Derivative
1998
·
Shuji Yonezawa
, Tadafumi Komurasaki
, et al.
·
The Journal of Organic Chemistry
·
42
Total Synthesis of Terprenin, a Highly Potent and Novel Immunoglobulin E Antibody Suppressant
1998
·
Kenji Kawada
, Akinori Arimura
, et al.
·
Angewandte Chemie International Edition
·
41
Synthesis and Antiviral Activity of 7-Benzyl-4-hydroxy-1,5-naphthyridin-2(1H)-one HIV Integrase Inhibitors
2009
·
Eric E. Boros
, Cynthia E. Edwards
, et al.
·
Journal of Medicinal Chemistry
·
40
Diastereoselective nucleophilic addition to chiral open-chain α-ketoacetals: Synthesis of (R)- and (S)-mevalolactone
1986
·
Yasumitsu Tamura
, Tomoko Ko
, et al.
·
Tetrahedron Letters
·
34
Asymmetric synthesis using chiral acetals: Highly diastereoselective addition of organocerium reagents to chiral .ALPHA.-aldoxime-ether acetal.
1989
·
Hiromichi FUJIOKA
, Masahiro FUJI
, et al.
·
Chemical and Pharmaceutical Bulletin
·
24
PDF
Asymmetric synthesis using chiral acetals: Studies on the nucleophilic addition of organometallics to chiral x-keto acetals in cyclic systems.
1987
·
YASUMITSU TAMURA
, HIROKAZU ANNOURA
, et al.
·
Chemical and Pharmaceutical Bulletin
·
19
PDF
Asymmetric synthesis using chiral acetals. Studies on the nucleophilic addition of organometallics to chiral .ALPHA.-keto acetals in open-chain systems.
1987
·
YASUMITSU TAMURA
, HIROKAZU ANNOURA
, et al.
·
Chemical and Pharmaceutical Bulletin
·
17
PDF
Asymmetric Synthesis of Carbapenems Using Chiral Acetals: Synthesis of a Key Intermediate to (+)-PS-5
1992
·
Hiromichi Fujioka
, Takeshi Yamanaka
, et al.
·
Synlett
·
12
A Stereoselective and Highly Practical Synthesis of Cytosolic Phospholipase A2 Substrate, 2-S-Arachidonoyl-1-O-hexadecyl-sn-2-thioglycero-3-O-phosphocholine
1997
·
Masahiro Fuji
, Fumihiko Watanabe,
, et al.
·
The Journal of Organic Chemistry
·
11
Totalsynthese von Terprenin, einem hochwirksamen Immunglobulin-E-Suppressivum
1998
·
Kenji Kawada
, Akinori Arimura
, et al.
·
Angewandte Chemie
·
9
Synthesis and Evaluation of Novel Nonpeptide Angiotensin II Receptor Antagonists: Imidazo(4,5-c)pyridine Derivatives with an Aromatic Substituent.
1995
·
Ryuichi KIYAMA
, Masahiro FUJI
, et al.
·
Chemical and Pharmaceutical Bulletin
·
9
PDF
Monomethylation of aromatic rings by Friedel-Crafts reaction with chloromethyl sulfide.
1986
·
YASUMITSU TAMURA
, HIROKAZU ANNOURA
, et al.
·
Chemical and Pharmaceutical Bulletin
·
8
PDF
The discovery of S/GSK1265744: a carbamoyl pyridone HIV‐1 integrase inhibitor
2012
·
Y Taoda
, B Johns
, et al.
·
Journal of the International AIDS Society
·
1
PDF
CCDC 935362: Experimental Crystal Structure Determination
2013
·
Johns, Brian A.
, Kawasuji, Takashi
, et al.
·
The Cambridge Structural Database
カルバモイルピリドン骨格を有する新規hivインテグラーゼ阻害薬の創製(1)リード化合物からドルテグラビルおよびs/gsk1265744への分子設計
2012
·
垰田善之
, A Johns Brian
, et al.
·
メディシナルケミストリーシンポジウム講演要旨集
カルバモイルピリドン骨格を有する新規hivインテグラーゼ阻害薬の創製(2)ジアステレオメリックアプローチによるドルテグラビルおよびs/gsk1265744の立体選択的合成研究
2012
·
秋山俊行
, A Johns Brian
, et al.
·
メディシナルケミストリーシンポジウム講演要旨集
3‐Hydroxy‐1,5‐dihydro‐pyrrol‐2‐one Derivatives (IV) as Advanced Inhibitors of HIV Integrase.
2007
·
Takashi Kawasuji
, Masahiro Fuji
, et al.
·
ChemInform
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Works count:
35
Citation count:
1,346
H-index:
15
I10-index:
17
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