Author

Hideyuki Kanno

Observed names: H. KANNO, H. Kanno, HIDEYUKI KANNO, Hideyuki KANNO

Observed institutions: Daiichi-Sankyo (Japan), Nihon Nohyaku (Japan), Weizmann Institute of Science, Teijin (Japan)

OpenAlex ID: A5113478814

Discovery of N-[(1R,2S,5S)-2-{[(5-chloroindol-2-yl)carbonyl]amino}-5-(dimethylcarbamoyl)cyclohexyl]-5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxamide hydrochloride: A novel, potent and orally active direct inhibitor of factor Xa

2008 · Tsutomu Nagata, Toshiharu Yoshino, et al. · Bioorganic & Medicinal Chemistry · 43

Cycloalkanediamine derivatives as novel blood coagulation factor Xa inhibitors

2007 · Tsutomu Nagata, Toshiharu Yoshino, et al. · Bioorganic & Medicinal Chemistry Letters · 33

Thromboxane A2 synthetase inhibitors. 2. Syntheses and activities of tetrahydronaphthalene and indane derivatives

1989 · Munefumi Kanao, Yoshifumi Watanabe, et al. · Journal of Medicinal Chemistry · 31

Synthesis and Antiallergy Activity of (1,3,4)Thiadiazolo(3,2-a)-1,2,3-triazolo(4,5-d)pyrimidin-9(3H)-one Derivatives. I.

1992 · Norio SUZUKI, Tamotsu MIWA, et al. · Chemical and Pharmaceutical Bulletin · 29

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New synthesis of (.+-.)-emetine from tetrahydroprotoberberine precursors via an .alpha.-diketone monothioketal intermediate

1978 · Seiichi Takano, Makoto Sasaki, et al. · The Journal of Organic Chemistry · 24

Facile Methods for Preparation of Thiazolopyridine and Tetrahydro-thiazolopyridine Derivatives

2004 · Noriyasu Haginoya, Satoshi Komoriya, et al. · Heterocycles · 22

An approach to a novel insect growth regulator buprofezin (Applaud)

1987 · H. Kanno · Pure and Applied Chemistry · 22

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Aryloxyacetic Acid Diuretics with Uricosuric Activity. II. Substituted ((4-Oxo-4H-1-benzopyran-7-yl)oxy)acetic Acids and the Related Compounds.

1991 · Masayuki KITAGAWA, Kenjiro YAMAMOTO, et al. · Chemical and Pharmaceutical Bulletin · 21

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Stereoselective synthesis and biological evaluation of 3,4-diaminocyclohexanecarboxylic acid derivatives as factor Xa inhibitors

2008 · Tsutomu Nagata, Masatoshi Nagamochi, et al. · Bioorganic & Medicinal Chemistry Letters · 16

Design, synthesis and SAR of novel ethylenediamine and phenylenediamine derivatives as factor Xa inhibitors

2011 · Kenji Yoshikawa, Toshiharu Yoshino, et al. · Bioorganic & Medicinal Chemistry Letters · 13

Diastereoselective Palladium(0)-catalyzed Reactions of Lithium Enolates of Chiral N-Acyloxazolidinones. Asymmetric Synthesis of 2-Substituted (E)-4-Alkylidenepentanedioates

1995 · Hideyuki Kanno, Ken Osanai · Tetrahedron Letters · 12

A Reagent, Ethyl 2-(2-tert-Butyl-2H-tetrazol-5-yl)-3-(dimethylamino)acrylate (DMTE), for Facile Synthesis of 2,3-(Ring Fused)-5-(5-teratzolyl)-4H-pyrimidin-4-one Derivatives.

1991 · Hideyuki KANNO, Hitoshi YAMAGUCHI, et al. · Chemical and Pharmaceutical Bulletin · 10

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Synthesis of (±)-Emetine from Protoberberine Precursor via the a-Diketone Monothioletal Intermediate

1977 · Seiichi Takano, Makoto Sasaki, et al. · Heterocycles · 10

2-Aminomethylphenylamine as a novel scaffold for factor Xa inhibitor

2011 · Akiyoshi Mochizuki, Tsutomu Nagata, et al. · Bioorganic & Medicinal Chemistry · 8

Diastereoselective addition-elimination reactions of lithium enolates of chiral N-acyloxazolidinones with 2-methylene-3-phenoxyalkanoates

1995 · Hideyuki Kanno, Ken Osanai · Tetrahedron Asymmetry · 8

Thromboxane A2 synthetase inhibitors. I. Syntheses and activities of various N-heteroaromatic derivatives.

1988 · MUNEFUMI KANAO, YOSHIFUMI WATANABE, et al. · Chemical and Pharmaceutical Bulletin · 5

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Orally active zwitterionic factor Xa inhibitors with long duration of action

2011 · Akiyoshi Mochizuki, Tsutomu Nagata, et al. · Bioorganic & Medicinal Chemistry Letters · 3

Potent inhibitors of neutral endopeptidase. 2-Biphenyl- methylglutaric acid amide derivatives

1996 · Hideyuki Kanno, Ken Osanai, et al. · Bioorganic & Medicinal Chemistry Letters · 3

Formation of 2,5-Dihydro-3H-pyrazolo[4,3-c]quinolin-3-ones from Ethyl 3-Amilino-2-(2-tert-butyl-2H-tetrazol-5-yl)acrylates

1992 · Sumiro Isoda, Hideyuki Kanno · Heterocycles · 3

Synthesis and Biological Activity of 1,3,5-thiadiazine Derivatives

1983 · K. Ikeda, H. Kanno, et al. · Elsevier eBooks · 3

Synthesis and evaluation of 2-(biphenylmethyl)glutaric acid amide derivatives as neutral endopeptidase inhibitors.

1996 · Hideyuki Kanno, Ken Osanai, et al. · Bioorganic & Medicinal Chemistry Letters · 1

ChemInform Abstract: A Facile Synthesis of 5,6‐Dihydro‐4H‐pyrrolo[3,4‐d]thiazole and Other Pyrrolidine‐Fused Aromatic Ring Systems via One‐Step Cyclization from Diols.

2012 · Kenji Yoshikawa, Tsutomu Nagata, et al. · ChemInform

ChemInform Abstract: Stereoselective Synthesis and Biological Evaluation of 3,4‐Diaminocyclohexanecarboxylic Acid Derivatives as Factor Xa Inhibitors.

2008 · Tsutomu Nagata, Masatoshi Nagamochi, et al. · ChemInform

Facile Methods for Preparation of Thiazolopyridine and Tetrahydrothiazolopyridine Derivatives.

2004 · Noriyasu Haginoya, Satoshi Komoriya, et al. · ChemInform

ChemInform Abstract: Potent Inhibitors of Neutral Endopeptidase. 2‐Biphenylmethylglutaric Acid Amide Derivatives.

1996 · H. KANNO, K. OSANAI, et al. · ChemInform

Works count: 38

Citation count: 320

H-index: 11

I10-index: 13