Author

Neil J. Press

Observed names: Neil J Press, Neil Press, Press, N.J., Press, Neil J.

Institutions: Novartis (Switzerland), Novartis Institutes for BioMedical Research

Observed institutions: Novartis (Switzerland), University of Sussex, University of Cambridge, Novartis (United Kingdom), Novartis Institutes for BioMedical Research, Imperial College London, University of Bath, The University of Texas at Austin

OpenAlex ID: A5113697483

Catalytic meta-selective C–H functionalization to construct quaternary carbon centres

2015 · Andrew J. Paterson, Sahra St John-Campbell, et al. · Chemical Communications · 173

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Dual PDE3/4 inhibitors as therapeutic agents for chronic obstructive pulmonary disease

2009 · Katharine H Banner, Neil J Press · British Journal of Pharmacology · 123

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An Inhibitor of NADPH Oxidase-4 Attenuates Established Pulmonary Fibrosis in a Rodent Disease Model

2013 · Elizabeth R. Jarman, Valerie S. Khambata, et al. · American Journal of Respiratory Cell and Molecular Biology · 114

Characterization of cigarette smoke-induced inflammatory and mucus hypersecretory changes in rat lung and the role of CXCR2 ligands in mediating this effect

2004 · Christopher S. Stevenson, Kevin Coote, et al. · American Journal of Physiology-Lung Cellular and Molecular Physiology · 90

2 PDE4 Inhibitors – A Review of the Current Field

2009 · Neil J. Press, Katharine H. Banner · Progress in medicinal chemistry · 61

Nitrone dipolar cycloaddition routes to piperidines and indolizidines. Part 9.Part 8. See Ref. 22. Formal synthesis of (–)-pinidine and total synthesis of (–)-histrionicotoxin, (+)-histrionicotoxin and (–)-histrionicotoxin 235AThis manuscript is dedicated to the sixtieth birthday of Professor L. Tietze.

2002 · Edwin C. Davison, Martin E. Fox, et al. · Journal of the Chemical Society Perkin Transactions 1 · 60

α-Halo carbonyls enable meta selective primary, secondary and tertiary C–H alkylations by ruthenium catalysis

2017 · Andrew J. Paterson, Callum J. Heron, et al. · Organic & Biomolecular Chemistry · 59

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The Crystalline Sponge Method: A Systematic Study of the Reproducibility of Simple Aromatic Molecule Encapsulation and Guest–Host Interactions

2016 · Lilian M. Hayes, Caroline E. Knapp, et al. · Crystal Growth & Design · 50

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Synthesis of a Protected (±)-Calicheamicinone Derivative by Sequential Introduction of Functionality into the Bicyclo[7.3.1]enediyne Core Structure

1997 · Philip Magnus, Gregory F. Miknis, et al. · Journal of the American Chemical Society · 36

Solubility-Driven Optimization of Phosphodiesterase-4 Inhibitors Leading to a Clinical Candidate

2012 · Neil J. Press, Roger J. Taylor, et al. · Journal of Medicinal Chemistry · 35

The total synthesis of alkaloids (–)-histrionicotoxin 259A, 285C and 285EAll new compounds exhibited satisfactory spectroscopic and analytical and/or exact mass data. Electronic supplementary information (ESI) available: experimental procedures for the preparation of compounds 4, 5, 13, 16, 22 and 25. See http://www.rsc.org/suppdata/cc/b1/b111514f/

2002 · Catherine J. Smith, Andrew B. Holmes, et al. · Chemical Communications · 34

A new orally bioavailable dual adenosine A2B/A3 receptor antagonist with therapeutic potential

2005 · Neil J. Press, Roger J. Taylor, et al. · Bioorganic & Medicinal Chemistry Letters · 31

Targeting the serotonin pathway for the treatment of pulmonary arterial hypertension

2013 · Matthew Thomas, Loredana Ciuclan, et al. · Pharmacology & Therapeutics · 29

Natural product drug delivery: A special challenge?

2019 · Neil J. Press, Emilie Joly, et al. · Progress in medicinal chemistry · 28

Therapeutic potential of adenosine receptor antagonists and agonists

2007 · Neil J Press, Stefania Gessi, et al. · Expert Opinion on Therapeutic Patents · 25

Intermolecular Interactions between Encapsulated Aromatic Compounds and the Host Framework of a Crystalline Sponge

2016 · Lilian M. Hayes, Neil J. Press, et al. · Crystal Growth & Design · 24

Microwave-Mediated Synthesis of an Arylboronate Library

2010 · John Spencer, Christine B. Baltus, et al. · ACS Combinatorial Science · 23

Discovery and Optimization of 4-(8-(3-Fluorophenyl)-1,7-naphthyridin-6-yl)transcyclohexanecarboxylic Acid, an Improved PDE4 Inhibitor for the Treatment of Chronic Obstructive Pulmonary Disease (COPD)

2015 · Neil J. Press, Roger J. Taylor, et al. · Journal of Medicinal Chemistry · 21

The discovery of potent, orally bioavailable pyrazolo and triazolopyrimidine CXCR2 receptor antagonists

2013 · David W. Porter, Michelle Bradley, et al. · Bioorganic & Medicinal Chemistry Letters · 21

The discovery of potent, orally bioavailable pyrimidine-5-carbonitrile-6-alkyl CXCR2 receptor antagonists

2014 · David W. Porter, Michelle Bradley, et al. · Bioorganic & Medicinal Chemistry Letters · 20

CGH2466, a combined adenosine receptor antagonist, p38 mitogen‐activated protein kinase and phosphodiesterase type 4 inhibitor with potent in vitro and in vivo anti‐inflammatory activities

2005 · Alexandre Trifilieff, Thomas H Keller, et al. · British Journal of Pharmacology · 20

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New Highly Potent and Selective Adenosine A3 Receptor Antagonists

2004 · Neil Press, Thomas Keller, et al. · Current Topics in Medicinal Chemistry · 20

Structure-based design and synthesis of phosphinate isosteres of phosphotyrosine for incorporation in Grb2-SH2 domain inhibitors. Part 1

2000 · Pascal Furet, Giorgio Caravatti, et al. · Bioorganic & Medicinal Chemistry Letters · 20

Intramolecular nitrone dipolar cycloadditions: control of regioselectivity and synthesis of naturally-occurring spirocyclic alkaloids

2012 · Alastair J. Hodges, Joseph P. Adams, et al. · Organic & Biomolecular Chemistry · 19

Efficient and Facile Synthesis of Acrylamide Libraries for Protein-Guided Tethering

2015 · Charlotte E. Allen, Peter R. Curran, et al. · Organic Letters · 18

Works count: 96

Citation count: 1,300

H-index: 20

I10-index: 32