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G. Griffiths

Observed name: Gary Griffiths
OpenAlex ID: A5113881172
2-Anilino-4-(thiazol-5-yl)pyrimidine CDK Inhibitors: Synthesis, SAR Analysis, X-ray Crystallography, and Biological Activity
2004 · Shudong Wang, Christopher Meades, et al. · Journal of Medicinal Chemistry · 153
Discovery and Characterization of 2-Anilino-4- (Thiazol-5-yl)Pyrimidine Transcriptional CDK Inhibitors as Anticancer Agents
2010 · Shudong Wang, Gary Griffiths, et al. · Chemistry & Biology · 107
Discovery ofN-Phenyl-4-(thiazol-5-yl)pyrimidin-2-amine Aurora Kinase Inhibitors
2010 · Shudong Wang, Carol A. Midgley, et al. · Journal of Medicinal Chemistry · 102
Synthesis and biological activity of 2-anilino-4-(1H-pyrrol-3-yl) pyrimidine CDK inhibitors
2004 · Shudong Wang, Gavin Wood, et al. · Bioorganic & Medicinal Chemistry Letters · 61
Insights into Cyclin Groove Recognition
2003 · George Kontopidis, Martin J.I. Andrews, et al. · Structure · 61
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Design, Synthesis, and Evaluation of 2-Methyl- and 2-Amino-N-aryl-4,5-dihydrothiazolo[4,5-h]quinazolin-8-amines as Ring-Constrained 2-Anilino-4-(thiazol-5-yl)pyrimidine Cyclin-Dependent Kinase Inhibitors
2010 · Neil A. McIntyre, Campbell McInnes, et al. · Journal of Medicinal Chemistry · 35
Cyclin A binding groove inhibitor Ace-Arg-Lys-Leu-Phe-Gly
2003 · G. Kontopidis, M. Andrews, et al. · Worldwide Protein Data Bank
Cyclin A binding groove inhibitor H-Cit-Cit-Leu-Ile-(p-F-Phe)-NH2
2003 · G. Kontopidis, M. Andrews, et al. · Worldwide Protein Data Bank
Cyclin A binding groove inhibitor Ac-Arg-Arg-Leu-Asn-(m-Cl-Phe)-NH2
2003 · G. Kontopidis, M. Andrews, et al. · Worldwide Protein Data Bank
Cyclin A binding groove inhibitor H-Ala-Ala-Abu-arg-er-Leu-Ile-(p-F-Phe)-NH2
2003 · G. Kontopidis, M. Andrews, et al. · Worldwide Protein Data Bank
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR N-[4-(2,4-Dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-N',N'-dimethyl-benzene-1,4-diamine
2003 · S. Wang, C. Meades, et al. · Worldwide Protein Data Bank
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR 4-[4-(4-Methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenol
2003 · S. Wang, C. Meades, et al. · Worldwide Protein Data Bank
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR [4-(2-Amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine
2003 · S. Wang, C. Meades, et al. · Worldwide Protein Data Bank
Works count: 15
Citation count: 520
H-index: 6
I10-index: 6
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