Get started
Author

Bert E. Thomas

Observed names: B. E. Thomas IV, Bert E Thomas, Bert E. Thomas IV, Bert Thomas
Observed institutions: Harvard University, University of California, Los Angeles, University of Pittsburgh, University of California, San Francisco, Sarcoma Foundation of America, Keymed Biosciences Inc. (China)
OpenAlex ID: A5115589595
Design and synthesis of sialyl Lewisx mimics as E‐ and P‐selectin inhibitors
2002 · Neelu Kaila, Bert E. Thomas IV · Medicinal Research Reviews · 95
Pharmacophore‐based molecular docking to account for ligand flexibility
2003 · Diane Joseph‐McCarthy, Bert E. Thomas, et al. · Proteins Structure Function and Bioinformatics · 80
Transition Structures of Thermally Allowed Disrotatory Electrocyclizations. The Prediction of Stereoselective Substituent Effects in Six-Electron Pericyclic Reactions
1995 · J. D. Evanseck, B. E. Thomas IV, et al. · The Journal of Organic Chemistry · 68
Secondary Kinetic Isotope Effects of Diastereotopic Protons in Pericyclic Reactions: A New Mechanistic Probe
1995 · Olaf Wiest, K. N. Houk, et al. · Journal of the American Chemical Society · 66
Design and synthesis of poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors. part 4: Biological evaluation of imidazobenzodiazepines as potent PARP-1 inhibitors for treatment of ischemic injuries
2003 · Dana Ferraris, Rica Pargas Ficco, et al. · Bioorganic & Medicinal Chemistry · 56
Electrocyclic reactions of 1-substituted 1,3,5,7-octatetraenes. An ab initio molecular orbital study of torquoselectivity in eight-electron electrocyclizations
1993 · Bert E. Thomas, J. D. Evanseck, et al. · Journal of the American Chemical Society · 49
Quinic Acid Derivatives as Sialyl Lewisx-Mimicking Selectin Inhibitors: Design, Synthesis, and Crystal Structure in Complex with E-Selectin
2005 · Neelu Kaila, William S. Somers, et al. · Journal of Medicinal Chemistry · 47
Transition Structures of the Ene Reactions of Cyclopropene
1997 · Qiaolin Deng, Bert E. Thomas, et al. · Journal of the American Chemical Society · 46
Torquoselectivity Induced by Lone-Pair Conjugation in the Electrocyclic Reactions of 1-Azapolyenes
2001 · Matthew J. Walker, Bruce N. Hietbrink, et al. · The Journal of Organic Chemistry · 40
Force field modeling of transition structures of intramolecular ene reactions and ab initio transition structures for an activated enophile
1992 · Bert E. Thomas, R. J. Loncharich, et al. · The Journal of Organic Chemistry · 40
Ketopyrrolidines and ketoazetidines as potent dipeptidyl peptidase IV (DPP IV) inhibitors
2004 · Dana Ferraris, Yao-Sen Ko, et al. · Bioorganic & Medicinal Chemistry Letters · 28
Synthesis, molecular modeling and biological evaluation of aza-proline and aza-pipecolic derivatives as FKBP12 ligands and their in vivo neuroprotective effects
2003 · Douglas E Wilkinson, Bert E Thomas, et al. · Bioorganic & Medicinal Chemistry · 25
An ab initio molecular orbital study of the first step of the catalytic mechanism of thymidylate synthase: the Michael addition of sulfur and oxygen nucleophiles
1995 · Bert E. Thomas, Peter A. Kollman · The Journal of Organic Chemistry · 25
Azetidine-Based Inhibitors of Dipeptidyl Peptidase IV (DPP IV)
2007 · Dana Ferraris, Sergei Belyakov, et al. · Current Topics in Medicinal Chemistry · 24
Design and synthesis of sialyl lewis x mimics as e-selectin inhibitors
2001 · Neelu Kaila, Bert E. Thomas, et al. · Bioorganic & Medicinal Chemistry Letters · 22
Insight into the specificity of thymidylate synthase from molecular dynamics and free energy perturbation calculations
1995 · Giulio Rastelli, Bert Thomas, et al. · Journal of the American Chemical Society · 17
Tuning exo/endo stereoselectivity in ene reactions
1993 · Bert E. Thomas, K. N. Houk · Journal of the American Chemical Society · 16
A Global Phase I Clinical Study Comparing the Safety and Pharmacokinetics of Proposed Biosimilar BAT1706 and Bevacizumab (Avastin®) in Healthy Male Subjects
2019 · Xiaoyun Wu, Chris Wynne, et al. · BioDrugs · 15
Synthesis and evaluation of chiral bicyclic proline FKBP12 ligands
2003 · David C. Limburg, Bert E. Thomas, et al. · Bioorganic & Medicinal Chemistry Letters · 15
Transition Structures of the Electrocyclic Reactions of cis,cis,cis‐1,3,5‐Cyclooctatriene
1993 · Bert E. Thomas, Jeffrey D. Evanseck, et al. · Israel Journal of Chemistry · 15
Selectin inhibitors
2003 · Neelu Kaila, Bert E Thomas · Expert Opinion on Therapeutic Patents · 11
Theoretical structures of methylenecyclopropane-2-carboxamide and related three-membered rings with exocyclic unsaturation. The origin of a ground-state distortion
1992 · Bert E. Thomas, K. N. Houk · The Journal of Organic Chemistry · 6
Abstract CT189: A phase I study of BAT1006, a novel anti-HER2 antibody, in patients with locally advanced/metastatic solid tumors
2023 · Xingxing Mei, Weijia Tang, et al. · Cancer Research
Sarcoma Patient Advocacy
2017 · Bert E. Thomas · Elsevier eBooks
List of Contributors
2017 · Siviero Agazzi, B. Aika Shoo, et al. · Elsevier eBooks
Works count: 26
Citation count: 806
H-index: 16
I10-index: 21
Year
Topic
Type