Keyword

indole functionalization

Description: Chemical modification of an indole ring or its substituents to introduce functional groups, principally in synthetic organic chemistry.

Primary topic: Synthesis of Indole Derivatives (37%)

OpenAlex ID: keywords/indole-functionalization

Synthesis and Functionalization of Indoles Through Palladium-catalyzed Reactions

2005 · Sandro Cacchi, Giancarlo Fabrizi · Chemical Reviews · 1,777

Update 1 of: Synthesis and Functionalization of Indoles Through Palladium-Catalyzed Reactions

2011 · Sandro Cacchi, Giancarlo Fabrizi · Chemical Reviews · 697

A Journey Across Recent Advances in Catalytic and Stereoselective Alkylation of Indoles

2005 · Marco Bandini, Achille Umani-Ronchi, et al. · Synlett · 371

Progress in palladium-based catalytic systems for the sustainable synthesis of annulated heterocycles: a focus on indole backbones

2012 · Mélanie Platon, Régine Amardeil, et al. · Chemical Society Reviews · 349

Transition Metals in the Synthesis and Functionalization of Indoles [New Synthesis Methods (72)]

1988 · Louis S. Hegedus · Angewandte Chemie International Edition in English · 344

Visible light-mediated chemistry of indoles and related heterocycles

2019 · Alexey A. Festa, Leonid G. Voskressensky, et al. · Chemical Society Reviews · 303

Synthesis of Cyclobutane-Fused Angular Tetracyclic Spiroindolines via Visible-Light-Promoted Intramolecular Dearomatization of Indole Derivatives

2019 · Min Zhu, Chao Zheng, et al. · Journal of the American Chemical Society · 299

Ir-Catalyzed Functionalization of 2-Substituted Indoles at the 7-Position: Nitrogen-Directed Aromatic Borylation

2006 · Sulagna Paul, Ghayoor A. Chotana, et al. · Journal of the American Chemical Society · 277

Recent Advances in Metal‐Catalyzed Functionalization of Indoles

2021 · Kelvin Urbina, David Tresp, et al. · Advanced Synthesis & Catalysis · 180

Aerobic Transition-Metal-Free Visible-Light Photoredox Indole C-3 Formylation Reaction

2014 · Xiang Li, Xiangyong Gu, et al. · ACS Catalysis · 156

Dual nickel and Lewis acid catalysis for cross-electrophile coupling: the allylation of aryl halides with allylic alcohols

2017 · Xue-Gong Jia, Peng Guo, et al. · Chemical Science · 139

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Visible-light-induced metal and reagent-free oxidative coupling of sp 2 C–H bonds with organo-dichalcogenides: synthesis of 3-organochalcogenyl indoles

2019 · Vandana Rathore, Sangit Kumar · Green Chemistry · 135

Indole Functionalization via Photoredox Gold Catalysis

2015 · Sherif J. Kaldas, Alexandre Cannillo, et al. · Organic Letters · 120

Copper-promoted decarboxylative direct C3-acylation of N-substituted indoles with α-oxocarboxylic acids

2013 · Lin Yu, Pinhua Li, et al. · Chemical Communications · 119

ZrCl4-Mediated Regio- and Chemoselective Friedel–Crafts Acylation of Indole

2011 · Sankar K. Guchhait, Maneesh Kashyap, et al. · The Journal of Organic Chemistry · 119

Highly Efficient Construction of Benzene Ring in Carbazoles by Palladium-Catalyzedendo-Mode Oxidative Cyclization of 3-(3‘-Alkenyl)indoles

2006 · Aidi Kong, Xiuling Han, et al. · Organic Letters · 118

Iridium‐Catalyzed Direct C4‐ and C7‐Selective Alkynylation of Indoles Using Sulfur‐Directing Groups

2019 · Chandrababu Naidu Kona, Yuji Nishii, et al. · Angewandte Chemie International Edition · 96

Electrochemically enabled chemoselective sulfonylation and hydrazination of indoles

2019 · Yu-Zhen Zhang, Zu-Yu Mo, et al. · Green Chemistry · 96

Palladium‐Catalyzed Direct Denitrogenative C‐3‐Arylation of 1H‐Indoles with Arylhydrazines using Air as the Oxidant

2013 · Yongxin Chen, Shuaibo Guo, et al. · Advanced Synthesis & Catalysis · 94

Unraveling the Structure and Reactivity Patterns of the Indole Radical Cation in Regioselective Electrochemical Oxidative Annulations

2023 · Xing Liu, Dali Yang, et al. · Journal of the American Chemical Society · 87

Direct Functionalization of Indoles: Copper-Catalyzed Malonyl Carbenoid Insertions

2010 · Michael B. Johansen, Michael A. Kerr · Organic Letters · 82

Indol-2-yltributylstannane: A Versatile Reagent for 2-Substituted Indoles

1994 · Sharada S. Labadie, Edmond Teng · The Journal of Organic Chemistry · 82

Pd(0)-Catalyzed Alkenylation and Allylic Dearomatization Reactions between Nucleophile-Bearing Indoles and Propargyl Carbonate

2014 · Run-Duo Gao, Chuan Liu, et al. · Organic Letters · 79

Multiple Roles of the Pyrimidyl Group in the Rhodium‐Catalyzed Regioselective Synthesis and Functionalization of Indole‐3‐carboxylic Acid Esters

2016 · Hui Jiang, Shang Gao, et al. · Advanced Synthesis & Catalysis · 78

Fused Heterocyclic Molecule-Functionalized N-Doped Reduced Graphene Oxide by Non-Covalent Bonds for High-Performance Supercapacitors

2020 · Liming Xu, Yingying Zhang, et al. · ACS Applied Materials & Interfaces · 77

Works count: 422

Citation count: 11,330