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2-Phenyl-9H-purine-6-carbonitrile derivatives as selective cathepsin S inhibitors

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Year: 2010
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2010.06.049
Authors: Jiaqiang Cai, D. Jonathan Bennett, Zoran Rankovic, Maureen Dempster, Xavier Fradera, Jonathan Gillespie, Iain Cumming, William Finlay, Mark Baugh, Sylviane Boucharens, John Bruin, Kenneth S. Cameron, William Hamilton, Jennifer Kerr, Emma Kinghorn, George McGarry, John Robinson, Paul Scullion, Joost C.M. Uitdehaag, Mario van Zeeland, Dominique Potin, Laurent Saniere, Andre Fouquet, Francois Chevallier, Hortense Deronzier, Cecile Dorleans, Eric Nicolai
Institutions: Merck B.V. (Netherlands), MSD (Netherlands)
Language: English

Topic: Protease and Inhibitor Mechanisms
Subfield: Cancer Research
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: closed
OpenAlex ID: W1992439997
FWCI: 0.987
Cites: 20
Cited by: 12
Related to: 10
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