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Pyrrolidine-pyrazole ureas as potent and selective inhibitors of 11β-hydroxysteroid-dehydrogenase type 1

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Year: 2011
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2011.02.111
Authors: Olivier Venier, Cécile Pascal, Alain Braun, Claudie Namane, Patrick Mougenot, Olivier Crespin, François Pacquet, Cécile Mougenot, Catherine Monseau, Bénédicte Onofri, Rommel Dadji-Faïhun, Céline Leger, Majdi Ben-Hassine, Thao Van-Pham, Jean-Luc Ragot, Christophe Philippo, Stefan Güssregen, Christian Engel, Géraldine Farjot, Lionel Noah, Karima Maniani, Eric Nicolaï
Institutions: Sanofi (France), Sanofi (Germany)
Language: English

Topic: Hormonal Regulation and Hypertension
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W1995769445
FWCI: 2.465
Cites: 37
Cited by: 15
Related to: 10
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