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Regioselective Glucuronidation of Andrographolide and Its Major Derivatives: Metabolite Identification, Isozyme Contribution, and Species Differences

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Year: 2014
Type: article
Source: The AAPS Journal
DOI: 10.1208/s12248-014-9658-8
Authors: Xiangge Tian, Sicheng Liang, Chao Wang, Baojian Wu, Guangbo Ge, Sa Deng, Kexin Liu, Ling Yang, Xiaochi Ma
Institutions: Dalian Medical University, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Jinzhou Medical University, Jinan University
Language: English

Topic: Pharmacogenetics and Drug Metabolism
Subfield: Pharmacology
Field: Pharmacology, Toxicology and Pharmaceutics
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: bronze

Funders: National Natural Science Foundation of China, Program for New Century Excellent Talents in University
Awards: G4739843997, G4989087030, 基于体内代谢特点的中药蟾酥中蟾蜍甾烯的结构与抗肿瘤活性、心脏毒性和代谢稳定性之间关系研究, G8826286050
OpenAlex ID: W1997758801
FWCI: 2.022
Cites: 40
Cited by: 35
Related to: 10
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