Discovery of (3 S ,3a R )-2-(3-Chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2 H -benzo[ g ]indazole-7-carboxylic Acid (PF-3882845), an Orally Efficacious Mineralocorticoid Receptor (MR) Antagonist for Hypertension and Nephropathy
Year: 2010
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/jm100505n
Authors: Marvin J. Meyers, Graciela B. Arhancet, Susan L. Hockerman, Xiangyang Chen, Scott A. Long, Matthew W. Mahoney, Joseph R. Rico, Danny J. Garland, James. R. Blinn, Joe T. Collins, Shengtian Yang, Horng-Chih Huang, Kevin F. McGee, Jay M. Wendling, Jessica D. Dietz, Maria A. Payne, Bruce L. Homer, Marcia I. Heron, David B. Reitz, Xiao Hu
Language: English
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
Open Access status: closed
OpenAlex ID: W2000625714
