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Structure–activity relationship study of acridine analogs as haspin and DYRK2 kinase inhibitors

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Year: 2010
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2010.04.150
Authors: Gregory D. Cuny, Maxime Robin, Natalia P. Ulyanova, Debasis Patnaik, Valerie Pique, Gilles Casano, Ji-Feng Liu, Xiangjie Lin, Jun Xian, Marcie A. Glicksman, Ross L. Stein, Jonathan M.G. Higgins
Institutions: Brigham and Women's Hospital, Harvard University, Centre National de la Recherche Scientifique, Aix-Marseille Université, Institut des Sciences Moléculaires de Marseille
Language: English

Topic: Heterocyclic Compound Synthesis and Bioactivity
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: green

Funder: National Cancer Institute
Award: Development of a haspin kinase assay for high throughput drug screening
OpenAlex ID: W2063532152
FWCI: 1.627
Cites: 24
Cited by: 62
Related to: 10
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