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Kinetic and structural characterization of caspase-3 and caspase-8 inhibition by a novel class of irreversible inhibitors

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Year: 2010
Type: article
Source: Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics
DOI: 10.1016/j.bbapap.2010.05.007
Authors: Zhigang Wang, William Watt, Nathan A. Brooks, Melissa S. Harris, Jan Urban, Douglas Boatman, Michael McMillan, Michael Kahn, Robert L. Heinrikson, Barry C. Finzel, Arthur J. Wittwer, James Blinn, Satwik Kamtekar, Alfredo G. Tomasselli
Institutions: Pfizer (United States), Arena Pharmaceuticals (United States), University of Southern California, Proteos (United States)
Language: English

Topic: Cell death mechanisms and regulation
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Institute of Microbiology, Chinese Academy of Sciences, Basic Energy Sciences
OpenAlex ID: W2141892423
FWCI: 1.04
Cites: 66
Cited by: 71
Related to: 10
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