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Discovery of potent, selective, and orally bioavailable quinoline-based dipeptidyl peptidase IV inhibitors targeting Lys554

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Year: 2011
Type: article
Source: Bioorganic & Medicinal Chemistry
DOI: 10.1016/j.bmc.2011.06.032
Authors: Hironobu Maezaki, Yoshihiro Banno, Yasufumi Miyamoto, Yuusuke Moritou, Tomoko Asakawa, Osamu Kataoka, Koji Takeuchi, Nobuhiro Suzuki, Koji Ikedo, Takuo Kosaka, Masako Sasaki, Shigetoshi Tsubotani, Akiyoshi Tani, Miyuki Funami, Yoshio Yamamoto, Michiko Tawada, Kathleen Aertgeerts, Jason Yano, Satoru Oi
Institution: Takeda (Japan)
Language: English

Topic: Diabetes Treatment and Management
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: U.S. Department of Energy, Basic Energy Sciences, Lawrence Berkeley National Laboratory
OpenAlex ID: W2149596087
FWCI: 1.026
Cites: 40
Cited by: 30
Related to: 10
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