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A novel potent metal-binding NDM-1 inhibitor was identified by fragment virtual, SPR and NMR screening

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Year: 2020
Type: article
Source: Bioorganic & Medicinal Chemistry
DOI: 10.1016/j.bmc.2020.115437
Authors: Huifang Guo, Kai Cheng, Yan Gao, Weiqi Bai, Cai Wu, Wei He, Conggang Li, Zhuorong Li
Institutions: Chinese Academy of Medical Sciences & Peking Union Medical College, Chinese Academy of Sciences, Wuhan Institute of Physics and Mathematics, Tsinghua University
Language: English

Topic: Antibiotic Resistance in Bacteria
Subfield: Microbiology (medical)
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: National Natural Science Foundation of China
Awards: 超级细菌中新型青霉素水解酶NDM-1动态构象的核磁共振波谱研究, G4799414056
OpenAlex ID: W3011980291
FWCI: 1.882
Cites: 48
Cited by: 22
Related to: 10
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