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N-Hydroxyformamide LpxC inhibitors, their in vivo efficacy in a mouse Escherichia coli infection model, and their safety in a rat hemodynamic assay

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Year: 2020
Type: article
Source: Bioorganic & Medicinal Chemistry
DOI: 10.1016/j.bmc.2020.115826
Authors: Takeru Furuya, Adam B. Shapiro, Janelle Comita-Prevoir, Eric J. Kuenstner, Jing Zhang, Seth D. Ribe, April Chen, Daniel Hines, Samir H. Moussa, Nicole M. Carter, Mark A. Sylvester, Jan A.C. Romero, Camilo V. Vega, Michael D. Sacco, Yu Chen, John P. O'Donnell, Thomas F. Durand-Reville, Alita A. Miller, Ruben A. Tommasi
Institutions: Entasis Therapeutics (United States), University of South Florida
Language: English

Topic: Synthesis and Biological Evaluation
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: bronze
OpenAlex ID: W3097315641
FWCI: 1.022
Cites: 34
Cited by: 23
Related to: 10
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