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Discovery of 1-Amino-1 H -imidazole-5-carboxamide Derivatives as Highly Selective, Covalent Bruton’s Tyrosine Kinase (BTK) Inhibitors

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Year: 2021
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.1c01559
Authors: Chunhua Ma, Qingyun Li, Minghao Zhao, Goujie Fan, Jie Zhao, Dandan Zhang, Shouning Yang, Shuting Zhang, Dingding Gao, Longfei Mao, Liang Zhu, Wei Li, Guiqing Xu, Yuqin Jiang, Qingjie Ding
Institutions: Henan Normal University, Shanghai University of Traditional Chinese Medicine
Language: English

Topic: Chronic Lymphocytic Leukemia Research
Subfield: Hematology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: National Natural Science Foundation of China
Awards: 靶向Toll样受体8的小分子抑制的设计合成、生物学评价及作用机制研究, G4510142828, G5408230873, G7641444476
OpenAlex ID: W3206073383
FWCI: 3.886
Cites: 26
Cited by: 42
Related to: 10
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