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A fragment-based drug discovery strategy applied to the identification of NDM-1 β-lactamase inhibitors

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Year: 2022
Type: article
Source: European Journal of Medicinal Chemistry
DOI: 10.1016/j.ejmech.2022.114599
Authors: Jérémy Caburet, Benjamin Boucherle, Sofiane Bourdillon, Giorgia Simoncelli, Federica Verdirosa, Jean-Denis Docquier, Yohann Moreau, Isabelle Krimm, Serge Crouzy, Marine Peuchmaur
Institutions: Centre National de la Recherche Scientifique, Commissariat à l'Énergie Atomique et aux Énergies Alternatives, Laboratoire de Chimie et Biologie des Métaux, Département de Pharmacochimie Moléculaire, Université Grenoble Alpes, University of Siena, University of Liège, Lyon 1 Université, Inserm, Centre Léon Bérard, Centre de Recherche en Cancérologie de Lyon
Language: English

Topic: Antibiotic Resistance in Bacteria
Subfield: Microbiology (medical)
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: bronze

Funders: LABoratoires d’EXcellence ARCANE, Agence Nationale de la Recherche
Awards: CBH-EUR-GS, G2389725886
OpenAlex ID: W4285037355
FWCI: 2.15
Cites: 56
Cited by: 19
Related to: 10
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