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Identification of reversible OATP1B1 and time-dependent CYP3A4 inhibition as the major risk factors for drug-induced cholestasis (DIC)

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Year: 2024
Type: article
Source: Archives of Toxicology
DOI: 10.1007/s00204-024-03794-3
Authors: Vlasia Kastrinou-Lampou, Raquel Rodríguez-Pérez, Birk Poller, Felix Huth, Zsuzsanna Gáborik, Beáta Mártonné-Tóth, Csilla Temesszentandrási-Ambrus, Heiko S. Schadt, Gerd A. Kullak-Ublick, Michael Arand, Gian Camenisch
Institutions: Novartis (Switzerland), University of Zurich, University Hospital Zurich
Language: English

Topic: Drug-Induced Hepatotoxicity and Protection
Subfield: Pharmacology
Field: Pharmacology, Toxicology and Pharmaceutics
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: green
OpenAlex ID: W4400780324
FWCI: 1.447
Cites: 39
Cited by: 6
Related to: 10
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