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Abstract 4378: BBO-11818, an orally bioavailable, highly potent and non-covalent pan-KRAS inhibitor demonstrates robust anti-tumor activity in KRAS-mutant preclinical models

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Year: 2025
Type: conference-abstract
Source: Cancer Research
DOI: 10.1158/1538-7445.am2025-4378
Authors: Carlos Ernesto Stahlhut Espinosa, Kanchan Singh, Zuhui Zhang, Kyle Sullivan, Nadege Gitego, Megan Rigby, Roger Ma, Patrick Alexander, Saman Setoodeh, Jin Shu, Ken Lin, Dana Rabara, Erik Larsen, Alok Sharma, Albert Chan, Brian P. Smith, Andrew Stephen, Yue Yang, Jun Pei, Felice C. Lightstone, Dhirendra Simanshu, Rui Xu, Chunmei Ji, Keshi Wang, Bin Wang, Kerstin Sinkevicius, Dwight V. Nissley, Eli Wallace, Frank McCormick, Anna E. Maciag, Pedro J. Beltran
Institutions: BridgeBio Oncology Therapeutics (United States), Frederick National Laboratory for Cancer Research, Lawrence Livermore National Laboratory
Language: English

Topic: Protein Kinase Regulation and GTPase Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W4409633147
Cites:
Cited by: 8
Related to: 10
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