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Discovery of INCB161734: A Selective Inhibitor of the KRAS G12D Mutant

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c02625
Authors: Alexander Sokolsky, Haolin Yin, Qinda Ye, Peter Carlsen, Chunyin Law, Matthew S. McCammant, Rocco Policarpo, Padmaja Polam, Le Zhao, Fenglei Zhang, Gencheng Li, Bin Hu, Wenyu Zhu, Gia Hoang, Robert Susick, Zhenwu Li, Pei Gan, Artem Shvartsbart, Jeremy J. Roach, Chao Qi, Sean Bowen, Chengtsung Lai, Abdellah Allali-Hassani, Keith Kennedy, Leslie B. Epling, Alexandra Gallion, Kerri Kurzeja-Lipinski, Karen Gallagher, Valerie Roman, Matthew R. Farren, Weixi Kong, Guofeng Zhang, Jason Boer, Marc C. Deller, Hui Wang, Maryanne Covington, Jennifer J. Harris, Sunkyu Kim, Dashyant Dhanak, Wenqing Yao, Xiaozhao Wang
Institution: Incyte (United States)
Language: English

Topic: Protein Kinase Regulation and GTPase Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: Incyte
OpenAlex ID: W7224842003
FWCI:
Cites: 44
Cited by:
Related to: 10
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