Discovery of INCB161734: A Selective Inhibitor of the KRAS G12D Mutant
Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
Authors: Alexander Sokolsky, Haolin Yin, Qinda Ye, Peter Carlsen, Chunyin Law, Matthew S. McCammant, Rocco Policarpo, Padmaja Polam, Le Zhao, Fenglei Zhang, Gencheng Li, Bin Hu, Wenyu Zhu, Gia Hoang, Robert Susick, Zhenwu Li, Pei Gan, Artem Shvartsbart, Jeremy J. Roach, Chao Qi, Sean Bowen, Chengtsung Lai, Abdellah Allali-Hassani, Keith Kennedy, Leslie B. Epling, Alexandra Gallion, Kerri Kurzeja-Lipinski, Karen Gallagher, Valerie Roman, Matthew R. Farren, Weixi Kong, Guofeng Zhang, Jason Boer, Marc C. Deller, Hui Wang, Maryanne Covington, Jennifer J. Harris, Sunkyu Kim, Dashyant Dhanak, Wenqing Yao, Xiaozhao Wang
Institution: Incyte (United States)
Language: English
Subfield: Molecular Biology
Domain: Life Sciences
Open Access status: closed
Funder: Incyte
OpenAlex ID: W7224842003
