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ABCB1, ABCG2, and CES1 are Key Determinants of the Pharmacokinetics of KRASG12C Inhibitor Divarasib

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Year: 2026
Type: article
Source: Molecular Pharmaceutics
DOI: 10.1021/acs.molpharmaceut.6c00463
Authors: Jamie Rijmers, Viët Bui, Daniëlle C. Band, Wenlong Li, Liesbeth Hoekman, Onno B. Bleijerveld, Davinia Arguedas, Olaf van Tellingen, Maria C. Lebre, Jos H. Beijnen, Alfred H. Schinkel
Institutions: The Netherlands Cancer Institute, University of Cambridge, Utrecht University
Language: English

Topic: Drug Transport and Resistance Mechanisms
Subfield: Oncology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W7225628016
FWCI:
Cites: 31
Cited by:
Related to: 10
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