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Robin Larouche‐Gauthier

Observed names: Larouche-Gauthier, R., Larouche-Gauthier, Robin, R. Larouche-Gauthier, Robin Larouche-Gauthier
ORCID: 0000-0003-1919-600X
Observed ORCID: 0000-0003-1919-600X
OpenAlex ID: A5007621532
Enantioselective Construction of Quaternary Stereogenic Centers from Tertiary Boronic Esters: Methodology and Applications
2011 · Ravindra P. Sonawane, Vishal Jheengut, et al. · Angewandte Chemie International Edition · 234
Ate Complexes of Secondary Boronic Esters as Chiral Organometallic-Type Nucleophiles for Asymmetric Synthesis
2011 · Robin Larouche-Gauthier, Tim G. Elford, et al. · Journal of the American Chemical Society · 204
Use of alkyl 2,4,6-triisopropylbenzoates in the asymmetric homologation of challenging boronic esters
2011 · Robin Larouche-Gauthier, Catherine J. Fletcher, et al. · Chemical Communications · 103
Enantioselective Construction of Quaternary Stereogenic Centers from Tertiary Boronic Esters: Methodology and Applications
2011 · Ravindra P. Sonawane, Vishal Jheengut, et al. · Angewandte Chemie · 75
Design of a brain-penetrant CDK4/6 inhibitor for glioblastoma
2019 · Sarah M. Bronner, Karl A. Merrick, et al. · Bioorganic & Medicinal Chemistry Letters · 73
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Intramolecular Additions of Various π-Nucleophiles to Chemoselectively Activated Amides and Application to the Synthesis of (±)-Tashiromine
2005 · Guillaume Bélanger, Robin Larouche-Gauthier, et al. · The Journal of Organic Chemistry · 70
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Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy
2021 · Jack A. Terrett, Huifen Chen, et al. · Journal of Medicinal Chemistry · 53
Rapid Assembly of Quinolizidines via Consecutive Nucleophilic Cyclizations onto Activated Amides
2011 · Guillaume Bélanger, Gary O’Brien, et al. · Organic Letters · 49
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Addition of Tethered Nonaromatic Carbon Nucleophiles to Chemoselectively Activated Amides
2005 · Guillaume Bélanger, Robin Larouche-Gauthier, et al. · Organic Letters · 42
Synthesis of the Tricyclic Core of Alkaloid Securinol B Using a Cascade of Vilsmeier−Haack and Mannich Cyclizations
2008 · Robin Larouche-Gauthier, Guillaume Bélanger · Organic Letters · 40
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Asymmetric Total Synthesis of (+)-Virosine A via Sequential Nucleophilic Cyclizations onto an Activated Formamide
2012 · Guillaume Bélanger, Marianne Dupuis, et al. · The Journal of Organic Chemistry · 36
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Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease
2024 · Jack A. Terrett, Justin Q. Ly, et al. · Journal of Medicinal Chemistry · 27
A Retrospective Look at the Impact of Binding Site Environment on the Optimization of TRPA1 Antagonists
2021 · Elisia Villemure, Jack A. Terrett, et al. · ACS Medicinal Chemistry Letters · 19
Optimization of a Novel DEL Hit That Binds in the Cbl-b SH2 Domain and Blocks Substrate Binding
2024 · Jun Liang, Michael J. Lambrecht, et al. · ACS Medicinal Chemistry Letters · 15
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Discovery of Selective Tertiary Amide Inhibitors of Cyclin-Dependent Kinase 2 (CDK2)
2023 · Mingshuo Zeng, Jessica M. Grandner, et al. · ACS Medicinal Chemistry Letters · 12
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Cp*Rh(III)‐Catalyzed C8 C−H Alkylation of Quinoline N‐Oxides with Diazo Meldrum's Acid
2021 · Malcolm P. Huestis, Jean‐Philippe Leclerc, et al. · European Journal of Organic Chemistry · 7
Prins cyclization of α-bromoethers under basic conditions
2013 · Patrice Arpin, Bryan Hill, et al. · Canadian Journal of Chemistry · 3
Optimization and In Vivo Characterization of a Series of Cbl-b Inactive-State Inhibitors
2026 · Michael J. Lambrecht, Jun Liang, et al. · ACS Medicinal Chemistry Letters · 1
Cover Picture: Enantioselective Construction of Quaternary Stereogenic Centers from Tertiary Boronic Esters: Methodology and Applications (Angew. Chem. Int. Ed. 16/2011)
2011 · Ravindra P. Sonawane, Vishal Jheengut, et al. · Angewandte Chemie International Edition · 1
Optimization Leading to a Potent and Selective Cbl-b Inactive-State Inhibitor That Demonstrated In Vivo Efficacy
2026 · Jun Liang, Michael J. Lambrecht, et al. · ACS Medicinal Chemistry Letters
Cover Feature: Cp*Rh(III)‐Catalyzed C8 C−H Alkylation of Quinoline N‐Oxides with Diazo Meldrum's Acid (Eur. J. Org. Chem. 3/2021)
2021 · Malcolm P. Huestis, Jean‐Philippe Leclerc, et al. · European Journal of Organic Chemistry
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CCDC 2048908: Experimental Crystal Structure Determination
2020 · Huestis, Malcolm P., Leclerc, Jean-Phillippe, et al. · The Cambridge Structural Database
ChemInform Abstract: Prins Cyclization of α‐Bromoethers under Basic Conditions.
2014 · Patrice Arpin, Bryan Hill, et al. · ChemInform
ChemInform Abstract: Use of Alkyl 2,4,6‐Triisopropylbenzoates in the Asymmetric Homologation of Challenging Boronic Esters.
2012 · Robin Larouche‐Gauthier, Catherine J. Fletcher, et al. · ChemInform
ChemInform Abstract: Enantioselective Construction of Quaternary Stereogenic Centers from Tertiary Boronic Esters: Methodology and Applications.
2011 · Ravindra P. Sonawane, Vishal Jheengut, et al. · ChemInform
Works count: 32
Citation count: 1,064
H-index: 14
I10-index: 15
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