Author

Maxim B. Nawrozkij

Observed names: Maxim Nawrozkij, Nawrozkij, Maxim B.

Institutions: Russian Academy of Sciences, Sirius University of Science and Technology, Institute of Physiologically Active Compounds

Observed institutions: Universitat Autònoma de Barcelona, Russian Academy of Sciences, University of Salerno, IrsiCaixa, Sirius University of Science and Technology, Istituto di Genetica Molecolare, Volgograd State Technical University, Hospital Universitari Germans Trias i Pujol, Istituto Pasteur, Institute of Physiologically Active Compounds, Sapienza University of Rome

ORCID: 0009-0003-5253-3706

Observed ORCID: 0009-0003-5253-3706

OpenAlex ID: A5113222123

Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains

2007 · Antonello Mai, Marino Artico, et al. · Journal of Medicinal Chemistry · 58

5-Alkyl-6-benzyl-2-(2-oxo-2-phenylethylsulfanyl)pyrimidin-4(3H)-ones, a Series of Anti-HIV-1 Agents of the Dihydro-alkoxy-benzyl-oxopyrimidine Family with Peculiar Structure−Activity Relationship Profile

2008 · Maxim B. Nawrozkij, Dante Rotili, et al. · Journal of Medicinal Chemistry · 56

Diarylpyrimidine−Dihydrobenzyloxopyrimidine Hybrids: New, Wide-Spectrum Anti-HIV-1 Agents Active at (Sub)-Nanomolar Level

2011 · Dante Rotili, Domenico Tarantino, et al. · Journal of Medicinal Chemistry · 53

1,2,4-Oxadiazoles in medicinal chemistry: trends of the last years

2025 · Anastasia Cherkasova, Roberta Astolfi, et al. · European Journal of Medicinal Chemistry · 38

2-(Alkyl/Aryl)Amino-6-Benzylpyrimidin-4(3H)-ones as Inhibitors of Wild-Type and Mutant HIV-1: Enantioselectivity Studies

2012 · Dante Rotili, Alberta Samuele, et al. · Journal of Medicinal Chemistry · 34

Effect of α-Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3H)-ones

2018 · Maxim B. Nawrozkij, Mariantonietta Forgione, et al. · Journal of Medicinal Chemistry · 26

Design, Synthesis, and Biological Evaluation of (+)‐Camphor‐ and (−)‐Fenchone‐Based Derivatives as Potent Orthopoxvirus Inhibitors

2022 · Anastasiya S. Sokolova, Kseniya S. Kovaleva, et al. · ChemMedChem · 25

Structural insight into the optimization of ethyl 5-hydroxybenzo[g]indol-3-carboxylates and their bioisosteric analogues as 5-LO/m-PGES-1 dual inhibitors able to suppress inflammation

2018 · Ferdinando Bruno, Suann Errico, et al. · European Journal of Medicinal Chemistry · 24

Exploring the Role of 2-Chloro-6-fluoro Substitution in 2-Alkylthio-6-benzyl-5-alkylpyrimidin-4(3H)-ones: Effects in HIV-1-Infected Cells and in HIV-1 Reverse Transcriptase Enzymes

2014 · Dante Rotili, Domenico Tarantino, et al. · Journal of Medicinal Chemistry · 24

Structure-Based Design, Synthesis, and Biological Evaluation of the Cage–Amide Derived Orthopox Virus Replication Inhibitors

2022 · Evgenii S. Mozhaitsev, Evgeniy V. Suslov, et al. · Viruses · 19

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Arbidol: a quarter-century after. Past, present and future of the original Russian antiviral

2017 · Konstantin V. Balakin, Rosanna Filosa, et al. · Russian Chemical Reviews · 19

Pyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity

2022 · Rossella Fioravanti, Eleonora Proia, et al. · European Journal of Medicinal Chemistry · 11

An Amazing 30-Year Journey around the DABO Family: A Medicinal Chemistry Lesson on a Versatile Class of Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

2025 · Emanuele Fabbrizi, Vladimir V. Chernyshov, et al. · Journal of Medicinal Chemistry · 8

(Heteroarylmethyl)benzoic Acids as a New Class of Bacterial Cystathionine γ-Lyase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling

2024 · Anastasia Golovina, Eleonora Proia, et al. · ACS Infectious Diseases · 4

A Practical Synthesis of 4’-Fluorospiro[cyclopropane-1,3’-indol]-2’(1’H)-one: a Valuable Terminal Building-Block for Biologically Active Podands

2016 · Alexandre S. Babushkin, Maxim B. Nawrozkij, et al. · Macroheterocycles · 2

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Convenient Synthesis of Building-Blocks for Pyridine/Piperidine-Decorated Crown Ethers

2014 · Maxim B. Nawrozkij, Evgeniy B. Gorbunov, et al. · Macroheterocycles · 1

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Systematic Structure–Activity Relationship Investigation on Novel 5-Alkyl-6-benzyl-2-{[(methylthio/phenylthio)alkyl]thio}-pyrimidin-4(3 H )-ones Endowed with Potent Anti-HIV-1 Activity

2026 · Gebremedhin Solomon Hailu, Egor Degtyarenko, et al. · ACS Omega

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Exploring the role of conformational restriction in 5-alkyl-6-benzyl-2-{[(methylthio)methyl]thio}pyrimidin-4(3H)-ones: Effects in HIV-1 infected cells and reverse transcriptase enzymes

2026 · Egor Degtyarenko, Gebremedhin Solomon Hailu, et al. · European Journal of Medicinal Chemistry

Comprehensive Risdiplam Synthesis Overview: From Cross-Coupling Reliance to Complete Palladium Independence

2025 · Georgiy Korenev, Maxim B. Nawrozkij, et al. · Molecules

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CCDC 2212428: Experimental Crystal Structure Determination