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Discovery of cyclic guanidines as potent, orally active, human glucagon receptor antagonists

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Year: 2011
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2011.09.085
Authors: Christopher Sinz, Jiang Chang, Ashley Rouse Lins, Ed Brady, Mari Candelore, Qing Dallas-Yang, Victor Ding, Guoqiang Jiang, Zhen Lin, Steven Mock, Sajjad Qureshi, Gino Salituro, Richard Saperstein, Jackie Shang, Deborah Szalkowski, Laurie Tota, Stella Vincent, Michael Wright, Shiyao Xu, Xiaodong Yang, Bei Zhang, James Tata, Ronald Kim, Emma Parmee
Institution: Merck & Co., Inc., Rahway, NJ, USA (United States)
Language: English

Topic: Diabetes Treatment and Management
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W1967494018
FWCI: 1.048
Cites: 14
Cited by: 9
Related to: 10
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