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Discovery of a novel competitive inhibitor of PTP1B by high-throughput screening

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Year: 2008
Type: article
Source: Acta Pharmacologica Sinica
DOI: 10.1111/j.1745-7254.2008.00737.x
Authors: Lei SHI, Hai-ping YU, Yue-yang ZHOU, Jun-qin DU, Qiang SHEN, Jing-ya LI, Jing-ya LI, Jia LI, Jia LI
Institutions: Chinese Academy of Sciences, Shanghai Institutes for Biological Sciences, Shanghai Institute of Materia Medica, National Center for Drug Screening
Language: English

Topic: Protein Tyrosine Phosphatases
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: National Natural Science Foundation of China
Awards: 蛋白酪氨酸磷酸酯酶1B选择性抑制剂在胰岛素敏感细胞内的作用机制研究, 结合传统中草药资源高通量筛选β-分泌酶抑制剂, 针对分子靶点的抗糖尿病药物发现及其机理研究
OpenAlex ID: W2010423744
FWCI: 2.357
Cites: 19
Cited by: 69
Related to: 10
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