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Discovery of Imine-Modified Quinazolinyl Sulfonamides as Dual hCA IX/XII Inhibitors with Potent Antiproliferative Activity

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Year: 2026
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.6c01358
Authors: Hazem Essam Okda, Lingaiah Maram, Mohammad Homaidur Rahman, Andrea Ammara, Simone Giovannuzzi, Dalia Kanaa, Hannah Duggan, Mohamed Elagawany, Lamees Hegazy, Claudiu T. Supuran, Bahaa Elgendy
Institutions: University of Health Sciences and Pharmacy, Washington University in St. Louis, University of Florence, American University in Cairo
Language: English

Topic: Enzyme function and inhibition
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W7165872445
FWCI: 1.857
Cites: 51
Cited by: 1
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