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Peter J. Webb

In Vitro and In Vivo Evaluation of APX001A/APX001 and Other Gwt1 Inhibitors against Cryptococcus
2018 · Karen Joy Shaw, Wiley A. Schell, et al. · Antimicrobial Agents and Chemotherapy · 127
3-(1 H -Tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole (MK-0354): A Partial Agonist of the Nicotinic Acid Receptor, G-Protein Coupled Receptor 109a, with Antilipolytic but No Vasodilatory Activity in Mice
2008 · Graeme Semple, Philip J. Skinner, et al. · Journal of Medicinal Chemistry · 104
1-Alkyl-benzotriazole-5-carboxylic Acids Are Highly Selective Agonists of the Human Orphan G-Protein-Coupled Receptor GPR109b
2006 · Graeme Semple, Philip J. Skinner, et al. · Journal of Medicinal Chemistry · 80
(1aR,5aR)1a,3,5,5a-Tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic Acid (MK-1903): A Potent GPR109a Agonist that Lowers Free Fatty Acids in Humans
2012 · P. Douglas Boatman, Brett Lauring, et al. · Journal of Medicinal Chemistry · 54
Fluorinated pyrazole acids are agonists of the high affinity niacin receptor GPR109a
2007 · Philip J. Skinner, Martin C. Cherrier, et al. · Bioorganic & Medicinal Chemistry Letters · 37
Potent tricyclic pyrazole tetrazole agonists of the nicotinic acid receptor (GPR109a)
2010 · P. Douglas Boatman, Thomas O. Schrader, et al. · Bioorganic & Medicinal Chemistry Letters · 34
Agonist lead identification for the high affinity niacin receptor GPR109a
2007 · Tawfik Gharbaoui, Philip J. Skinner, et al. · Bioorganic & Medicinal Chemistry Letters · 31
3-Nitro-4-amino benzoic acids and 6-amino nicotinic acids are highly selective agonists of GPR109b
2007 · Philip J. Skinner, Martin C. Cherrier, et al. · Bioorganic & Medicinal Chemistry Letters · 30
A calcineurin antifungal strategy with analogs of FK506
2017 · Mitchell Nambu, Jonathan A. Covel, et al. · Bioorganic & Medicinal Chemistry Letters · 28
Synthesis of analogs of the Gwt1 inhibitor manogepix (APX001A) and in vitro evaluation against Cryptococcus spp
2019 · Michael Trzoss, Jonathan A. Covel, et al. · Bioorganic & Medicinal Chemistry Letters · 27
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5-N,N-Disubstituted 5-aminopyrazole-3-carboxylic acids are highly potent agonists of GPR109b
2009 · Philip J. Skinner, Peter J. Webb, et al. · Bioorganic & Medicinal Chemistry Letters · 25
A versatile route to benzocanthinones
2005 · J. Hodge Markgraf, Adrian A. Dowst, et al. · Tetrahedron · 25
Solid-Phase Organic Synthesis and Combinatorial Chemistry: A Laboratory Preparation of Oligopeptides
2002 · George A. Truran, Karelle S. Aiken, et al. · Journal of Chemical Education · 15
The Discovery of Manogepix/Fosmanogepix and Other Gwt1 Inhibitors for the Treatment of Invasive Fungal Infections
2019 · Jonathan A. Covel, Quinlyn A. Soltow, et al. · Medicinal chemistry reviews · 7
A Versatile Route to Benzocanthinones.
2005 · J. Hodge Markgraf, Adrian A. Dowst, et al. · ChemInform · 1
A Versatile Synthesis of Benzacanthinones by Intramolecular Radical Coupling
2005 · J. Markgraf, A. Dowst, et al. · Synfacts
Works count: 16
Citation count: 624
H-index: 13
I10-index: 13
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