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Potent tricyclic pyrazole tetrazole agonists of the nicotinic acid receptor (GPR109a)

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Year: 2010
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2010.03.062
Authors: P. Douglas Boatman, Thomas O. Schrader, Michelle Kasem, Benjamin R. Johnson, Philip J. Skinner, Jae-Kyu Jung, Jerry Xu, Martin C. Cherrier, Peter J. Webb, Graeme Semple, Carleton R. Sage, Jens Knudsen, Ruoping Chen, Andrew K. Taggart, Ester Carballo-Jane, Jeremy G. Richman
Institutions: Arena Pharmaceuticals (United States), Merck & Co., Inc., Rahway, NJ, USA (United States)
Language: English

Topic: Heterocyclic Compound Synthesis and Bioactivity
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W1982134384
FWCI: 2.218
Cites: 18
Cited by: 34
Related to: 10
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