Author

Daryl A. Scherzer

Observed names: D. Scherzer, Daryl Scherzer

Institution: GlaxoSmithKline (United States)

Observed institution: GlaxoSmithKline (United States)

OpenAlex ID: A5079017404

Identification of Potent, Selective, Cell-Active Inhibitors of the Histone Lysine Methyltransferase EZH2

2012 · Sharad K. Verma, Xinrong Tian, et al. · ACS Medicinal Chemistry Letters · 390

Structure-Based Design of Potent and Selective 3-Phosphoinositide-Dependent Kinase-1 (PDK1) Inhibitors

2011 · Jesús R. Medina, Christopher J. Becker, et al. · Journal of Medicinal Chemistry · 56

Discovery of potent, selective sulfonylfuran urea endothelial lipase inhibitors

2008 · Krista B. Goodman, Michael J. Bury, et al. · Bioorganic & Medicinal Chemistry Letters · 53

Abstract 2939: Discovery and synthesis of highly potent and selective small molecule inhibitors of the histone methyltransferase EZH2

2012 · Sharad K. Verma, Louis V. LaFrance, et al. · Cancer Research · 1

Phosphoinositide-Dependent Kinase-1 (PDK1) kinase domain with 6-(3-Amino-1H-indazol-6-yl)-N4-ethyl-2,4-pyrimidinediamine

2011 · J.R. Medina, C.J. Becker, et al. · Worldwide Protein Data Bank

Phosphoinositide-Dependent Kinase-1 (PDK1) kinase domain with 4-[2-Amino-6-(3-amino-1H-indazol-6-yl)-4-pyrimidinyl]-N-phenyl-2-morpholinecarboxamide

2011 · J.R. Medina, C.J. Becker, et al. · Worldwide Protein Data Bank

Phosphoinositide-Dependent Kinase-1 (PDK1) kinase domain with 1,1-Dimethylethyl {(3R,6S)-1-[2-amino-6-(3-amino-1H-indazol-6-yl)-4-pyrimidinyl]-6-methyl-3-piperidinyl}carbamate

2011 · J.R. Medina, C.J. Becker, et al. · Worldwide Protein Data Bank

Works count: 9

Citation count: 500

H-index: 3

I10-index: 3