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Structure-Based Design of Potent and Selective 3-Phosphoinositide-Dependent Kinase-1 (PDK1) Inhibitors

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Year: 2011
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/jm101527u
Authors: Jesús R. Medina, Christopher J. Becker, Charles W. Blackledge, Celine Duquenne, Yanhong Feng, Seth W. Grant, Dirk Heerding, William H. Li, William H. Miller, Stuart P. Romeril, Daryl Scherzer, Arthur Shu, Mark A. Bobko, Antony R. Chadderton, Melissa Dumble, Christine M. Gardiner, Seth Gilbert, Qi Liu, Sridhar K. Rabindran, Valery Sudakin, Hong Xiang, Pat G. Brady, Nino Campobasso, Paris Ward, Jeffrey M. Axten
Institution: GlaxoSmithKline (United States)
Language: English

Topic: PI3K/AKT/mTOR signaling in cancer
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2017544644
FWCI: 2.033
Cites: 32
Cited by: 56
Related to: 10
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